SCHEMBL21582003

SCHEMBL21582003

CCn1nc(Br)cc1[N+](=O)[O-]

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.38
RAB9A P51151 1/20 0.36
ALDH1A1 P00352 4/20 0.35
LMNA P02545 2/20 0.35
THRB P10828 1/20 0.35
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
MAPT P10636 1/20 0.34
POLB P06746 2/20 0.33
MEN1 O00255 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
KMT2A Q03164 1/20 0.33
HTT P42858 1/20 0.33
GLA P06280 1/20 0.33
PDE4A P27815 1/20 0.32
PDE4B Q07343 1/20 0.32
PDE4C Q08493 1/20 0.32
PDE4D Q08499 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28435272 0.79 ALDH1A1 (0.39) SMN1; SMN2RAB9AALDH1A1LMNAMAPT
SCHEMBL21291535 0.76 CHEK1 (0.39) SMN1; SMN2ALDH1A1LMNATHRBTSHR
SCHEMBL28394145 0.75 DGAT1 (0.35) LMNAKMT2A
SCHEMBL5813872 0.72 PDE4A (0.41) SMN1; SMN2RAB9AALDH1A1LMNAMAPT
SCHEMBL20528938 0.72 KMT2A (0.40) SMN1; SMN2RAB9AALDH1A1LMNAMAPT
SCHEMBL4388002 0.72 MAPK1 (0.34) ALDH1A1LMNATHRBTSHRMAPK1
SCHEMBL18717726 0.70
SCHEMBL21582005 0.69 ADORA2A (0.36) MAPT
SCHEMBL19098523 0.67 ALDH1A1 (0.36) SMN1; SMN2RAB9AALDH1A1LMNATHRB
SCHEMBL30625835 0.67 SMN1; SMN2 (0.40) SMN1; SMN2ALDH1A1LMNATHRBTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3728257-A1 AUTOTAXIN INHIBITORS AND USES THEREOF Fronthera U.S. Pharmaceuticals LLC (US) 2020-10-28 EP disclosed
WO-2019228403-A1 AUTOTAXIN INHIBITORS AND USES THEREOF FRONTHERA U.S. PHARMACEUTICALS LLC (US) 2019-12-05 WO disclosed