SCHEMBL21590177

SCHEMBL21590177

Cc1cccc(Cl)c1NC(=O)c1ccccc1

nearest known ligand 0.77

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LCK P06239 3/20 0.68
LMNA P02545 2/20 0.64
KMT2A Q03164 2/20 0.64
MEN1 O00255 1/20 0.64
POLB P06746 2/20 0.57
HPGD P15428 1/20 0.57
TYK2 P29597 1/20 0.57
CHRNA7 P36544 1/20 0.56
MAPK14 Q16539 1/20 0.54
MAOB P27338 1/20 0.53
MAPT P10636 1/20 0.53
PDK1 Q15118 1/20 0.52
PDK2 Q15119 1/20 0.52
PDK3 Q15120 1/20 0.52
PDK4 Q16654 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1437928 0.88 KMT2A (0.80) LMNAKMT2AMEN1HPGDTYK2
SCHEMBL4138460 0.88 POLB (0.67) LCKLMNAKMT2AMEN1POLB
SCHEMBL21590301 0.86 MEN1 (0.55) LCKLMNAKMT2AMEN1TYK2
SCHEMBL11402399 0.84 PDK1 (0.59) LCKKMT2APOLBCHRNA7MAPK14
SCHEMBL28510576 0.83 LCK (0.61) LCKLMNAKMT2AMEN1TYK2
SCHEMBL7827455 0.83 POLB (0.79) LCKKMT2AMEN1POLBCHRNA7
SCHEMBL773400 0.83 LCK (1.00) LCKLMNACHRNA7MAPT
SCHEMBL773593 0.83 LCK (1.00) LCKMAPK14
SCHEMBL3785470 0.81 LMNA (0.66) LMNAKMT2AMEN1POLBHPGD
SCHEMBL18610497 0.81 RORC (0.63) LCKLMNAKMT2AMEN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111635404-B Preparation method of duloxetine 苏州明锐医药科技有限公司 2023-11-07 CN claimed
CN-111675710-B Preparation method of duloxetine 上海奥萝拉医药科技有限公司 2023-08-18 CN claimed
CN-111675710-A Preparation method of dovinisine 苏州明锐医药科技有限公司 2020-09-18 CN claimed
CN-111635404-A Preparation method of dovinisine 苏州明锐医药科技有限公司 2020-09-08 CN claimed
CN-118388485-B Du Weili Sibub synthesis method 江苏海洋大学 2024-11-05 CN disclosed
CN-118388485-A Du Weili Sibub synthesis method 江苏海洋大学 2024-07-26 CN disclosed
CN-118324765-A Synthesis method of PI3K inhibitor Du Weili sibutra 江苏海洋大学 2024-07-12 CN disclosed
CN-111635404-B Preparation method of duloxetine 苏州明锐医药科技有限公司 2023-11-07 CN disclosed
CN-111675710-B Preparation method of duloxetine 上海奥萝拉医药科技有限公司 2023-08-18 CN disclosed
CN-111675710-A Preparation method of dovinisine 苏州明锐医药科技有限公司 2020-09-18 CN disclosed
CN-111635404-A Preparation method of dovinisine 苏州明锐医药科技有限公司 2020-09-08 CN disclosed
WO-2019238067-A1 PYRROLO [2, 3-B] PYRIDINES OR PYRROLO [2, 3-B] PYRAZINES AS HPK1 INHIBITOR AND THE USE THEREOF BEIGENE, LTD. (KY) 2019-12-19 WO disclosed
CN-109071462-A Quinazoline derivative or salt thereof and pharmaceutical composition containing the same 柳韩洋行 2018-12-21 CN disclosed
CN-104447727-B Substituted amino-metadiazine compound and its application method and purposes 广东东阳光药业有限公司 2018-04-27 CN disclosed
CN-107690433-A Heteroaryl derivative or its pharmaceutically acceptable salt, its preparation method and include the pharmaceutical composition for being used to prevent or treat PI3 kinase-associated conditions ited as active component 韩国化学研究院 2018-02-13 CN disclosed
CN-104447727-A Substituted aminopyrimidine compound as well as use method and application thereof GUANGDONG HEC PHARMACEUTICAL 2015-03-25 CN disclosed