SCHEMBL21598835

SCHEMBL21598835

N#Cc1csc2c1CCNCC2

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.42
HTR2C P28335 2/20 0.42
HTR2B P41595 2/20 0.42
PNMT P11086 4/20 0.39
DRD2 P14416 2/20 0.30
DRD3 P35462 2/20 0.30
APEX1 P27695 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15848407 0.87 PNMT (0.41) HTR2AHTR2CHTR2BPNMTDRD2
SCHEMBL15920403 0.78 BPTF (0.41)
SCHEMBL21598840 0.77 PNMT (0.39) PNMTDRD2DRD3APEX1
SCHEMBL18430366 0.76 ALDH1A1 (0.43)
SCHEMBL2991516 0.72 HTR2C (0.41) HTR2AHTR2CHTR2BPNMT
SCHEMBL2996134 0.72 PNMT (0.36) HTR2AHTR2CHTR2BPNMTAPEX1
SCHEMBL25364670 0.68
SCHEMBL25365128 0.66 ADRA1A (0.34) DRD2DRD3
Hydrochloric Acid SCHEMBL31564391 0.65 NR2E1 (0.33)
SCHEMBL17377146 0.64 PNMT (0.45) PNMTAPEX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3810613-A1 N-SUBSTITUTED TETRAHYDROTHIENOPYRIDINE DERIVATIVES AND USES THEREOF Novartis AG (CH) 2021-04-28 EP disclosed
WO-2019244047-A1 N-SUBSTITUTED TETRAHYDROTHIENOPYRIDINE DERIVATIVES AND USES THEREOF NOVARTIS AG (CH) 2019-12-26 WO disclosed