SCHEMBL21606405

SCHEMBL21606405

CCOC(=O)c1cn(-c2ncc(Br)cc2OC)cn1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.49
OPRK1 P41145 6/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
DPP4 P27487 3/20 0.37
ALDH1A1 P00352 3/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2C19 P33261 1/20 0.37
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
THRB P10828 1/20 0.36
GABRG2 P18507 1/20 0.36
GABRB3 P28472 1/20 0.36
GABRA5 P31644 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
PDGFRB P09619 1/20 0.35
PDGFRA P16234 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21606397 0.89 NOTUM (0.47) NOTUMOPRK1MEN1KMT2AALDH1A1
SCHEMBL21606347 0.79 GABRA2 (0.42) OPRK1ALDH1A1GAAMAPTTHRB
SCHEMBL195517 0.77 PSEN1 (0.42)
SCHEMBL27592203 0.76 NOTUM (0.53) NOTUMMEN1KMT2AALDH1A1CYP1A2
SCHEMBL9372779 0.75 NOTUM (0.61) NOTUMMEN1KMT2A
SCHEMBL9465006 0.75 NOTUM (0.68) NOTUMMEN1KMT2AGAAMAPT
SCHEMBL21639372 0.74 NOTUM (0.67) NOTUMMEN1KMT2AALDH1A1CYP1A2
SCHEMBL21195187 0.73 MEN1 (0.33) MEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL1881082 0.72 NOTUM (0.65) NOTUMMEN1KMT2AALDH1A1CYP1A2
SCHEMBL21606545 0.71 RORC (0.42) OPRK1ALDH1A1GAAMAPTTHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019244000-A1 PHENYL AND PYRIDINYL SUBSTITUTED IMIDAZOLES AS MODULATORS OF RORYT JANSSEN PHARMACEUTICA NV (BE) 2019-12-26 WO disclosed