SCHEMBL21606765

SCHEMBL21606765

COc1ccc(C(c2ccccc2)(c2ccc(OC)cc2)N2C(=O)NC3C(CCCCC(=O)O)SCC32)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 5/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
MAPK1 P28482 2/20 0.42
MEN1 O00255 1/20 0.42
ABL1 P00519 1/20 0.42
LMNA P02545 1/20 0.42
PKM P14618 1/20 0.42
IDE P14735 1/20 0.42
KMT2A Q03164 1/20 0.42
RIN1 Q13671 1/20 0.42
KEAP1 Q14145 1/20 0.38
CA12 O43570 2/20 0.37
CA1 P00915 2/20 0.37
CA2 P00918 2/20 0.37
CA9 Q16790 2/20 0.37
CYP2J2 P51589 1/20 0.35
PDE4B Q07343 1/20 0.34
PTGFR P43088 1/20 0.34
GAA P10253 1/20 0.34
LTB4R Q15722 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30205123 1.00 TDP1 (0.42) TDP1L3MBTL1MAPK1MEN1ABL1
SCHEMBL30331593 1.00 TDP1 (0.42) TDP1L3MBTL1MAPK1MEN1ABL1
SCHEMBL23812201 0.93 TDP1 (0.47) TDP1L3MBTL1MAPK1MEN1ABL1
SCHEMBL16478559 0.93 TDP1 (0.47) TDP1L3MBTL1MAPK1MEN1ABL1
SCHEMBL16141184 0.90 HLCS (0.39) TDP1MEN1KMT2AKEAP1CA12
SCHEMBL30929050 0.84 HSP90AB1 (0.43) PKMKEAP1
SCHEMBL30929049 0.84 HSP90AB1 (0.43) PKMKEAP1
SCHEMBL9971307 0.83 KEAP1 (0.40) TDP1KEAP1ALDH1A1
SCHEMBL30205084 0.82 KEAP1 (0.40) TDP1KEAP1ALDH1A1
SCHEMBL21606770 0.78 CYP2J2 (0.32) TDP1L3MBTL1MAPK1MEN1ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019243273-A1 GOLD (I)-PHOSPHINE 1,2,3-TRIAZOLE DERIVATIVES WITH ANTIOBIOTIC PROPERTIES UNIVERSITÉ DE STRASBOURG (FR) 2019-12-26 WO disclosed