SCHEMBL21616640

SCHEMBL21616640

CCOC[C@@H]1CC(c2ccc(C(F)(F)F)cc2)CN1c1ccc(C#N)cc1

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.38
ELANE P08246 9/20 0.37
CYP2C9 P11712 3/20 0.37
HSD11B1 P28845 1/20 0.36
CYP3A4 P08684 5/20 0.36
HTT P42858 1/20 0.36
DGKZ Q13574 1/20 0.35
HRH3 Q9Y5N1 1/20 0.34
HTR2C P28335 1/20 0.33
AR P10275 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23632253 0.91 HSD11B1 (0.40) KIF11ELANECYP2C9HSD11B1CYP3A4
SCHEMBL28537013 0.89 ELANE (0.36) KIF11ELANECYP2C9HSD11B1CYP3A4
SCHEMBL28532578 0.88 KIF11 (0.37) KIF11ELANECYP2C9HSD11B1CYP3A4
SCHEMBL21616650 0.88 KIF11 (0.37) KIF11HSD11B1CYP3A4HTTHRH3
SCHEMBL21616677 0.86 KIF11 (0.37) KIF11ELANECYP2C9HSD11B1CYP3A4
SCHEMBL21616587 0.85 KIF11 (0.42) KIF11ELANECYP2C9HSD11B1CYP3A4
SCHEMBL21616599 0.84 KIF11 (0.41) KIF11ELANECYP2C9HSD11B1CYP3A4
SCHEMBL28526814 0.83 SRD5A2 (0.39)
SCHEMBL23633001 0.83 EPHX2 (0.43) KIF11DGKZHRH3
SCHEMBL28535402 0.82 HSD11B1 (0.38) KIF11ELANECYP2C9HSD11B1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112513021-B ROR gamma antagonist and application thereof in medicines 广东东阳光药业有限公司 2023-06-27 CN disclosed
CN-112513021-A ROR gamma antagonist and application thereof in medicine 广东东阳光药业有限公司 2021-03-16 CN disclosed
WO-2020011147-A1 RORγ ANTAGONIST AND APPLICATION THEREOF IN MEDICINE SUNSHINE LAKE PHARMA CO., LTD. (CN) 2020-01-16 WO disclosed