SCHEMBL28537013

SCHEMBL28537013

COCCOC[C@@H]1CC(c2ccc(C(F)(F)F)cc2)CN1c1ccc(C#N)cc1

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ELANE P08246 7/20 0.36
CYP3A4 P08684 3/20 0.36
HTT P42858 1/20 0.36
KIF11 P52732 1/20 0.36
FASN P49327 4/20 0.35
HSD11B1 P28845 1/20 0.35
CYP2C9 P11712 3/20 0.33
USP30 Q70CQ3 1/20 0.33
P2RY14 Q15391 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28532578 0.90 KIF11 (0.37) ELANECYP3A4HTTKIF11HSD11B1
SCHEMBL21616640 0.89 KIF11 (0.38) ELANECYP3A4HTTKIF11HSD11B1
SCHEMBL21616650 0.86 KIF11 (0.37) CYP3A4HTTKIF11FASNHSD11B1
SCHEMBL28533648 0.84 P2RY14 (0.43) HTTP2RY14
SCHEMBL21616677 0.84 KIF11 (0.37) ELANECYP3A4HTTKIF11HSD11B1
SCHEMBL21616587 0.83 KIF11 (0.42) ELANECYP3A4HTTKIF11HSD11B1
SCHEMBL21616599 0.82 KIF11 (0.41) ELANECYP3A4HTTKIF11HSD11B1
SCHEMBL28535402 0.81 HSD11B1 (0.38) ELANECYP3A4HTTKIF11FASN
SCHEMBL28535429 0.81 HSD11B1 (0.37) ELANECYP3A4HTTKIF11FASN
SCHEMBL23632253 0.80 HSD11B1 (0.40) ELANECYP3A4HTTKIF11HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112513021-B ROR gamma antagonist and application thereof in medicines 广东东阳光药业有限公司 2023-06-27 CN disclosed
CN-112513021-A ROR gamma antagonist and application thereof in medicine 广东东阳光药业有限公司 2021-03-16 CN disclosed