SCHEMBL23632253

SCHEMBL23632253

CCOCC1CCC(c2ccc(C(F)(F)F)cc2)CN1c1ccc(C#N)cc1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.40
KIF11 P52732 1/20 0.37
ELANE P08246 5/20 0.37
CYP2C9 P11712 2/20 0.37
HRH3 Q9Y5N1 2/20 0.36
CYP3A4 P08684 5/20 0.35
HTR2C P28335 2/20 0.35
HTT P42858 1/20 0.35
DGKZ Q13574 1/20 0.34
P2RY14 Q15391 1/20 0.34
EPHX2 P34913 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28535402 0.91 HSD11B1 (0.38) HSD11B1KIF11ELANECYP2C9HRH3
SCHEMBL21616640 0.91 KIF11 (0.38) HSD11B1KIF11ELANECYP2C9HRH3
SCHEMBL28537768 0.90 HSD11B1 (0.38) HSD11B1KIF11HRH3CYP3A4HTR2C
SCHEMBL28535429 0.89 HSD11B1 (0.37) HSD11B1KIF11ELANECYP2C9CYP3A4
SCHEMBL30474464 0.87 KDM1A (0.35) KIF11HTR2CDGKZ
SCHEMBL28540005 0.86 KIF11 (0.41) HSD11B1KIF11ELANECYP2C9HRH3
SCHEMBL21616615 0.85 HSD11B1 (0.42) HSD11B1KIF11CYP3A4HTR2CHTT
SCHEMBL23632362 0.85 HSD11B1 (0.42) HSD11B1KIF11CYP3A4HTR2CHTT
SCHEMBL28539964 0.84 HSD11B1 (0.42) HSD11B1KIF11ELANECYP2C9HRH3
SCHEMBL21616645 0.84 P2RY14 (0.38) P2RY14EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113072542-B ROR gamma t inhibitor and preparation method and application thereof 广东东阳光药业股份有限公司 2024-04-05 CN disclosed
WO-2021139595-A1 RORγT INHIBITOR, PREPARATION METHOD THEREFOR AND USE THEREOF 东莞市东阳光新药研发有限公司 2021-07-15 WO disclosed
CN-113072542-A ROR gamma t inhibitor and preparation method and application thereof 广东东阳光药业有限公司 2021-07-06 CN disclosed