SCHEMBL21621707

SCHEMBL21621707

CCOC(=O)c1nc(C)n(-c2cccc(C(=O)OC)c2C)c1C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.50
RAB9A P51151 2/20 0.50
POLB P06746 1/20 0.50
MYC P01106 1/20 0.46
TSHR P16473 2/20 0.45
CYP1A2 P05177 1/20 0.40
TP53 P04637 3/20 0.40
CDC25A P30304 1/20 0.40
CDC25B P30305 1/20 0.40
CDC25C P30307 1/20 0.40
THRB P10828 1/20 0.40
MAPT P10636 2/20 0.39
GAA P10253 1/20 0.39
KMT2A Q03164 1/20 0.39
KDM4E B2RXH2 1/20 0.39
ELANE P08246 1/20 0.39
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
SLC6A4 P31645 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4965866 0.78 PDE4A (0.45) RAB9ATSHRCYP1A2TP53MAPT
SCHEMBL16935806 0.78 SLC5A1 (0.49) ALDH1A1RAB9APOLBTSHRCYP1A2
SCHEMBL20763779 0.74 TSHR (0.66) ALDH1A1TSHRCYP1A2CDC25ACDC25B
SCHEMBL1078509 0.74 TP53 (0.58) ALDH1A1RAB9ATP53MAPTGAA
SCHEMBL1708108 0.74 POLB (0.53) ALDH1A1RAB9APOLBMYCTSHR
SCHEMBL4958802 0.73 ALDH1A1 (0.57) ALDH1A1CYP1A2TP53THRBMAPT
SCHEMBL18355727 0.73 ALDH1A1 (0.51) ALDH1A1POLBCYP1A2TP53ELANE
SCHEMBL18355722 0.73 ALDH1A1 (0.60) ALDH1A1POLBTP53KMT2AELANE
SCHEMBL21621661 0.72 GABRG2 (0.47) ALDH1A1TSHR
SCHEMBL1707968 0.71 TSHR (0.47) ALDH1A1RAB9APOLBMYCTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020011246-A1 BENZENE RING-CONTAINING COMPOUND, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF 广州丹康医药生物有限公司 2020-01-16 WO disclosed