SCHEMBL21636760

SCHEMBL21636760

COC(=N)c1cccc(Br)c1C

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 6/20 0.35
MEN1 O00255 4/20 0.35
AHR P35869 1/20 0.35
ALDH1A1 P00352 4/20 0.34
HPGD P15428 2/20 0.34
HSD17B10 Q99714 1/20 0.34
KDM4E B2RXH2 3/20 0.33
MAPT P10636 2/20 0.33
F2R P25116 1/20 0.33
MIF P14174 1/20 0.33
POLB P06746 1/20 0.33
GAA P10253 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22308161 0.85 ALDH1A1 (0.33) NPC1RAB9AKMT2AALDH1A1HPGD
SCHEMBL21842993 0.81 F2R (0.40) NPC1RAB9AKMT2AMEN1ALDH1A1
SCHEMBL22307186 0.80 F2R (0.33) NPC1RAB9AKMT2AMEN1AHR
SCHEMBL22307183 0.80 ALDH1A1 (0.31) ALDH1A1CYP2C19
SCHEMBL25119548 0.79 MIF (0.39) NPC1RAB9AKMT2AMEN1AHR
SCHEMBL2134095 0.78 SMN1; SMN2 (0.37) NPC1RAB9AKMT2AMEN1ALDH1A1
SCHEMBL257409 0.77 LMNA (0.50) RAB9AKMT2AMEN1ALDH1A1HSD17B10
SCHEMBL30280732 0.77 LMNA (0.50) RAB9AKMT2AMEN1ALDH1A1HSD17B10
SCHEMBL4509521 0.76 C1S (0.39) ALDH1A1HPGDHSD17B10MAPTMIF
SCHEMBL30906644 0.74 NPC1 (0.40) NPC1RAB9AKMT2AMEN1AHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022022600-A1 IMMUNOMODULATORS, COMPOSITIONS AND METHODS THEREOF BETTA PHARMACEUTICALS CO., LTD (CN) 2022-02-03 WO disclosed
WO-2020156323-A1 IMMUNOMODULATORS, COMPOSITIONS AND METHODS THEREOF BETTA PHARMACEUTICALS CO., LTD (CN) 2020-08-06 WO disclosed
WO-2020015717-A1 IMMUNOMODULATORS, COMPOSITIONS AND METHODS THEREOF BETTA PHARMACEUTICALS CO., LTD (CN) 2020-01-23 WO disclosed