SCHEMBL21646360

SCHEMBL21646360

CSNc1ccn2cncc2c1

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PRKCI P41743 1/20 0.39
TBXAS1 P24557 1/20 0.38
BRD4 O60885 1/20 0.32
CREBBP Q92793 1/20 0.32
NR3C1 P04150 1/20 0.31
NAMPT P43490 1/20 0.31
NTRK1 P04629 1/20 0.31
IDO1 P14902 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23055267 0.77 PRKCI (0.39) PRKCITBXAS1BRD4CREBBPNR3C1
SCHEMBL25124500 0.77 TBXAS1 (0.40) PRKCITBXAS1BRD4CREBBPNR3C1
SCHEMBL21646352 0.70 MAPK1 (0.36)
SCHEMBL23697851 0.70 ESR1 (0.31)
SCHEMBL24629446 0.69 TBXAS1 (0.43) PRKCITBXAS1NR3C1NAMPTNTRK1
SCHEMBL15246478 0.67 TBXAS1 (0.43) PRKCITBXAS1BRD4CREBBPNR3C1
SCHEMBL17561679 0.67 TBXAS1 (0.40) PRKCITBXAS1BRD4CREBBPNR3C1
SCHEMBL13931946 0.67 QPCT (0.43) PRKCITBXAS1BRD4CREBBP
SCHEMBL15435640 0.67 TBXAS1 (0.54) PRKCITBXAS1BRD4CREBBPNR3C1
SCHEMBL31646996 0.65 LMNA (0.39) PRKCITBXAS1NAMPTNTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020017587-A1 PYRIDAZINONE DERIVATIVE 大日本住友製薬株式会社 2020-01-23 WO disclosed