SCHEMBL21652270

SCHEMBL21652270

c1ccc(-c2ccccc2NCC(Nc2ccccn2)c2ccccc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.55
HTT P42858 1/20 0.55
NPSR1 Q6W5P4 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
CYP2D6 P10635 1/20 0.46
CHRNB2 P17787 1/20 0.40
CHRNB4 P30926 1/20 0.40
CHRNA3 P32297 1/20 0.40
CHRNA4 P43681 1/20 0.40
ALDH1A1 P00352 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ADRA2A P08913 1/20 0.39
ADRA2B P18089 1/20 0.39
ADRA2C P18825 1/20 0.39
MAOA P21397 1/20 0.39
ADRA1D P25100 1/20 0.39
MAOB P27338 1/20 0.39
ADRA1A P35348 1/20 0.39
MEN1 O00255 1/20 0.38
MAPK10 P53779 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21652176 0.78 SLC10A1 (0.49) KDM4EHTTNPSR1L3MBTL1CYP2D6
SCHEMBL6420641 0.75 KDM4E (0.69) KDM4EHTTNPSR1L3MBTL1CYP2D6
SCHEMBL6754929 0.75 KDM4E (0.69) KDM4EHTTNPSR1L3MBTL1CYP2D6
SCHEMBL6564769 0.72 KDM4E (0.69) KDM4EHTTNPSR1L3MBTL1CYP2D6
SCHEMBL16805225 0.72 MEN1 (0.68) KDM4ECHRNB2CHRNB4CHRNA3CHRNA4
Hydrochloric Acid SCHEMBL6302647 0.71 KDM4E (0.67) KDM4EHTTNPSR1L3MBTL1CYP2D6
SCHEMBL21652279 0.71 SLC10A1 (0.45) KDM4EHTTNPSR1L3MBTL1CYP2D6
SCHEMBL21652272 0.70 SLC10A1 (0.44) KDM4EHTTNPSR1L3MBTL1CYP2D6
SCHEMBL21652166 0.69 ALDH1A1 (0.43) KDM4EHTTL3MBTL1CHRNB2CHRNA4
SCHEMBL4281005 0.67 CYP2D6 (0.72) KDM4EHTTNPSR1L3MBTL1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020019911-A1 BORON NITROGEN LIGAND BASED ON CHIRAL 1,2-ETHYLENEDIAMINE BACKBONE AND PREPARATION METHOD AND USE THEREOF 中国科学院兰州化学物理研究所苏州研究院 2020-01-30 WO disclosed