SCHEMBL21670367

SCHEMBL21670367

O=C(Nc1cccc(Cl)c1F)[C@H]1CCCNC1

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TNKS O95271 1/20 0.58
TNKS2 Q9H2K2 1/20 0.58
ROCK2 O75116 3/20 0.54
HTR6 P50406 2/20 0.47
CD274 Q9NZQ7 1/20 0.46
CDK9 P50750 4/20 0.45
CCNT1 O60563 1/20 0.44
PARP1 P09874 1/20 0.44
CXCR2 P25025 3/20 0.44
PBK Q96KB5 1/20 0.44
ULK1 O75385 1/20 0.43
F10 P00742 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21669972 0.86 TNKS (0.57) TNKSTNKS2ROCK2HTR6CD274
SCHEMBL2447263 0.83 TNKS (0.58) TNKSTNKS2ROCK2HTR6CD274
SCHEMBL22591708 0.78 MEN1 (0.62)
SCHEMBL4755192 0.77 SLC6A2 (0.49)
SCHEMBL2451469 0.77 TNKS (0.58) TNKSTNKS2ROCK2HTR6CD274
Hydrochloric Acid SCHEMBL16670883 0.77 TNKS (0.46) TNKSTNKS2ROCK2HTR6CD274
SCHEMBL21669919 0.76 ULK1 (0.56) ROCK2CDK9CCNT1ULK1F10
SCHEMBL21669936 0.76 ULK1 (0.56) ROCK2CDK9CCNT1ULK1F10
SCHEMBL2449231 0.75 F10 (0.56) TNKSTNKS2ULK1F10
SCHEMBL2452221 0.75 F10 (0.56) TNKSTNKS2ULK1F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020028482-A1 SMALL MOLECULES THAT SENSITIZE HIV-1 INFECTED CELLS TO ANTIBODY DEPENDENT CELLULAR CYTOTOXICITY THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2020-02-06 WO disclosed