SCHEMBL4755192

SCHEMBL4755192

O=C(c1cccc(Cl)c1F)C1CCCNC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 11/20 0.49
SLC6A4 P31645 11/20 0.49
SLC6A3 Q01959 11/20 0.49
KCNH2 Q12809 6/20 0.46
CHRM1 P11229 1/20 0.43
SLC6A1 P30531 2/20 0.42
SLC6A11 P48066 1/20 0.42
TSHR P16473 1/20 0.42
LMNA P02545 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
SLC6A13 Q9NSD5 1/20 0.42
KDM4E B2RXH2 1/20 0.41
MAPT P10636 1/20 0.41
KMT2A Q03164 1/20 0.41
ATM Q13315 1/20 0.41
CYP2D6 P10635 1/20 0.41
P2RX7 Q99572 1/20 0.41
OPRK1 P41145 1/20 0.40
KAT7 O95251 1/20 0.40
KAT6A Q92794 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9017801 0.87 SLC6A2 (0.55) SLC6A2SLC6A4SLC6A3KCNH2SLC6A1
SCHEMBL4779495 0.86 SLC6A1 (0.42) SLC6A2SLC6A4SLC6A3KCNH2SLC6A1
SCHEMBL26599052 0.84 KDM2B (0.46) SLC6A2SLC6A4SLC6A3CHRM1TSHR
SCHEMBL30606587 0.84 KDM2B (0.46) SLC6A2SLC6A4SLC6A3CHRM1TSHR
SCHEMBL21670367 0.77 TNKS (0.58)
SCHEMBL13631069 0.76 KMT2A (0.38) SLC6A2SLC6A4SLC6A3KCNH2SLC6A1
SCHEMBL26085824 0.75 KDM4E (0.49) SLC6A1SLC6A11TSHRLMNASMN1; SMN2
SCHEMBL4748847 0.75 KAT7 (0.44) SLC6A2SLC6A4SLC6A3KCNH2OPRK1
SCHEMBL4776325 0.74 SLC6A2 (0.41) SLC6A2SLC6A4SLC6A3KCNH2SLC6A1
SCHEMBL3963692 0.73 KDM2B (0.55) LMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008156832-A2 RENIN INHIBITORS VITAE PHARMACEUTICALS, INC. (US) 2008-12-24 WO disclosed
WO-2007117560-A2 PIPERIDINE AND MORPHOLINE RENIN INHIBITORS VITAE PHARMACEUTICALS, INC. (US) 2007-10-18 WO disclosed