SCHEMBL21676598

SCHEMBL21676598

CCC(C)(C)OC(=O)N[C@H](Cc1ccc(C#N)cc1)C(=O)NC1CCN(C)CC1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 2/20 0.46
CHRM3 P20309 6/20 0.45
CHRM2 P08172 1/20 0.45
CTSS P25774 6/20 0.43
CTSK P43235 5/20 0.43
SCN9A Q15858 2/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
SSTR4 P31391 1/20 0.42
CTSL P07711 1/20 0.42
CTSB P07858 1/20 0.42
DRD2 P14416 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21169918 0.92 CTSS (0.52) PIN1CHRM3CHRM2CTSSCTSK
SCHEMBL7983717 0.82 CTSS (0.55) CHRM3CHRM2CTSSCTSKSCN9A
SCHEMBL7983723 0.82 CTSS (0.55) CHRM3CHRM2CTSSCTSKSCN9A
SCHEMBL3054407 0.79 SCN9A (0.64) CTSSCTSKSCN9AKDM4ECTSL
SCHEMBL18930225 0.76 DPP4 (0.52) PIN1CHRM3CHRM2SSTR4DRD2
Hydrochloric Acid SCHEMBL21144960 0.75 DPP4 (0.51) PIN1CHRM3CHRM2SSTR4DRD2
Hydrochloric Acid SCHEMBL21144961 0.75 DPP4 (0.51) PIN1CHRM3CHRM2SSTR4DRD2
SCHEMBL22338765 0.74 P2RX7 (0.57) CTSSCTSKCTSLCTSB
SCHEMBL22303692 0.74 P2RX7 (0.57) CTSSCTSKCTSLCTSB
SCHEMBL21144825 0.73 CTSL (0.55) CTSSCTSKSCN9ACTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3383865-B1 FURANE DERIVATIVES AS INHIBITORS OF ATAD2 Bayer Pharma AG (DE) 2020-01-29 EP disclosed