SCHEMBL21697653

SCHEMBL21697653

Cc1c(Cc2cc3ccccc3s2)cc(Br)c(OCc2ccccc2)c1C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 3/20 0.40
AGXT P21549 1/20 0.40
ADRB2 P07550 1/20 0.40
THRA P10827 2/20 0.38
THRB P10828 2/20 0.38
ASIC3 Q9UHC3 1/20 0.37
LOXL2 Q9Y4K0 1/20 0.37
IDH1 O75874 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
CTRC Q99895 1/20 0.35
ADRA1D P25100 2/20 0.35
CHRNA7 P36544 1/20 0.34
HTR1D P28221 1/20 0.34
HTR1B P28222 1/20 0.34
SLC5A2 P31639 1/20 0.34
SENP5 Q96HI0 1/20 0.34
SENP2 Q9HC62 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16020862 0.84 CYP2A6 (0.40) CYP2A6AGXTADRB2THRATHRB
SCHEMBL21697576 0.83 CYP2A6 (0.37) CYP2A6AGXTADRB2THRATHRB
SCHEMBL20741882 0.82 CYP2A6 (0.40) CYP2A6AGXTADRB2ASIC3LOXL2
SCHEMBL16018686 0.80 CYP2A6 (0.50) CYP2A6AGXTADRB2ASIC3LOXL2
SCHEMBL20741835 0.79 SLC5A2 (0.44) CYP2A6AGXTADRB2SLC5A2
SCHEMBL21697633 0.77 SLC5A2 (0.40) CYP2A6AGXTADRB2ASIC3LOXL2
SCHEMBL21697598 0.77 SLC5A2 (0.42) CYP2A6AGXTADRB2ASIC3LOXL2
SCHEMBL21697652 0.77 THRB (0.38) THRATHRBSMN1; SMN2GAAMAPT
SCHEMBL28202032 0.75 CYP2A6 (0.50) CYP2A6AGXTADRB2ASIC3LOXL2
SCHEMBL21697640 0.74 AGXT (0.40) CYP2A6AGXTADRB2ADRA1DCHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2968258-B1 DUAL SGLT1/SGLT2 INHIBITORS JANSSEN PHARMACEUTICA NV (BE) 2020-02-12 EP disclosed