SCHEMBL21701575

SCHEMBL21701575

COc1ccc(C(=O)N(C)c2ccc(N3CCC(c4cccc(C)c4)C3)cc2C(=O)O)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MYC P01106 3/20 0.43
ALDH1A1 P00352 6/20 0.40
LMNA P02545 3/20 0.40
HPGD P15428 1/20 0.40
HIF1A Q16665 1/20 0.40
PDE5A O76074 1/20 0.40
DPP4 P27487 1/20 0.39
MALT1 Q9UDY8 1/20 0.39
NOTUM Q6P988 1/20 0.39
MAPT P10636 4/20 0.38
MAPK1 P28482 2/20 0.38
KDM4E B2RXH2 1/20 0.38
GAA P10253 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
HSD11B1 P28845 1/20 0.38
RAB9A P51151 4/20 0.37
NPC1 O15118 3/20 0.37
TP53 P04637 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21701596 0.78 SMN1; SMN2 (0.44) ALDH1A1HPGDMAPTKDM4EGAA
SCHEMBL21701582 0.77 KEAP1 (0.46) ALDH1A1MAPTKDM4ETDP1L3MBTL1
SCHEMBL21701416 0.67 MALT1 (0.81) ALDH1A1LMNAMALT1MAPTGAA
SCHEMBL31284692 0.66 TDP1 (0.45) ALDH1A1LMNAHPGDMALT1NOTUM
SCHEMBL21701422 0.66 MALT1 (0.67) ALDH1A1LMNAHPGDMALT1MAPT
SCHEMBL6677639 0.64 LMNA (0.60) ALDH1A1LMNAMAPTKDM4EL3MBTL1
SCHEMBL6677642 0.64 LMNA (0.60) ALDH1A1LMNAMAPTKDM4EL3MBTL1
SCHEMBL2943952 0.64 USP2 (0.56) ALDH1A1LMNANOTUMMAPTKDM4E
SCHEMBL31284461 0.63 NOTUM (0.56) ALDH1A1HPGDMALT1NOTUMMAPT
SCHEMBL12529764 0.63 MCHR1 (0.61)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020033944-A2 NON-POLYAMINE BASED POLYAMINE TRANSPORT INHIBITORS AND THEIR USE IN THE TREATMENT OF HUMAN CANCERS UNIVERSITY OF CENTRAL FLORIDA RESEARCH FOUNDATION, INC. (US) 2020-02-13 WO disclosed