SCHEMBL2170202

SCHEMBL2170202

COC(CC(=O)N1CCCC1C(N)=O)c1ccc(Oc2ccc(F)cc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 4/20 0.49
DPP4 P27487 3/20 0.48
HTR1A P08908 3/20 0.46
HTR7 P34969 3/20 0.46
FPR2 P25090 2/20 0.43
DPP8 Q6V1X1 2/20 0.42
DPP7 Q9UHL4 2/20 0.42
KMT2A Q03164 1/20 0.41
KCNH2 Q12809 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20575743 0.85 DPP4 (0.49) DPP4HTR1AHTR7
SCHEMBL2355316 0.82 SCN9A (0.52) SCN9ADPP4HTR1AHTR7FPR2
SCHEMBL2170169 0.75 SCN9A (0.54) SCN9ADPP4FPR2
SCHEMBL2356691 0.74 SCN9A (0.48) SCN9ADPP4HTR1AHTR7FPR2
SCHEMBL20575304 0.74 DPP4 (0.47) DPP4HTR1AHTR7
SCHEMBL12836594 0.74 LGMN (0.45) DPP4
SCHEMBL12895270 0.73 F2 (0.45) DPP4
SCHEMBL12463762 0.72 DPP4 (0.56) SCN9ADPP4HTR1AHTR7FPR2
SCHEMBL2172455 0.71 SCN9A (0.60) SCN9ADPP4HTR1AHTR7FPR2
SCHEMBL2170987 0.71 CYP2C9 (0.50) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346821-A1 SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS Exelixis, Inc. (US) 2011-07-27 EP disclosed