SCHEMBL2170169

SCHEMBL2170169

NC(=O)C1CCCN1C(=O)C(c1ccccc1)c1ccc(Oc2ccc(F)cc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 3/20 0.54
AGTR2 P50052 14/20 0.46
FPR2 P25090 1/20 0.46
RAB9A P51151 1/20 0.44
DPP4 P27487 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6980126 0.87 AGTR2 (0.52) AGTR2DPP4
SCHEMBL2171155 0.86 SCN9A (0.52) SCN9AFPR2RAB9ADPP4
SCHEMBL2355316 0.82 SCN9A (0.52) SCN9AFPR2RAB9ADPP4
SCHEMBL2356691 0.79 SCN9A (0.48) SCN9AFPR2RAB9ADPP4
SCHEMBL2352727 0.77 SCN9A (0.53) SCN9AFPR2DPP4
SCHEMBL31376320 0.76 DPP4 (0.65) RAB9ADPP4
SCHEMBL13570514 0.76 F2 (0.53) RAB9ADPP4
SCHEMBL2170202 0.75 SCN9A (0.49) SCN9AFPR2DPP4
SCHEMBL2176481 0.74 KCNH2 (0.47) RAB9ADPP4
SCHEMBL2172455 0.73 SCN9A (0.60) SCN9AFPR2DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2349252-A2 SYNERGISTIC COMBINATION OF SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS AND ANTIMICROTUBULE AGENTS Exelixis, Inc. (US) 2011-08-03 EP disclosed
EP-2346821-A1 SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS Exelixis, Inc. (US) 2011-07-27 EP disclosed