SCHEMBL2356691

SCHEMBL2356691

NC(=O)C1CCCN1C(=O)C(c1ccc(Oc2ccc(F)cc2)cc1)N1CCOCC1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 7/20 0.48
FPR2 P25090 5/20 0.45
HTR1A P08908 1/20 0.41
HTR7 P34969 1/20 0.41
DPP4 P27487 1/20 0.40
KCNK3 O14649 3/20 0.40
ALDH1A1 P00352 1/20 0.40
TSHR P16473 1/20 0.39
HTT P42858 1/20 0.39
RAB9A P51151 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C19 P33261 1/20 0.38
KCNH2 Q12809 1/20 0.37
LMNA P02545 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
APOL1 O14791 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2170169 0.79 SCN9A (0.54) SCN9AFPR2DPP4RAB9A
SCHEMBL2355316 0.79 SCN9A (0.52) SCN9AFPR2HTR1AHTR7DPP4
SCHEMBL2170202 0.74 SCN9A (0.49) SCN9AFPR2HTR1AHTR7DPP4
SCHEMBL3733552 0.74 LMNA (0.52) DPP4ALDH1A1TSHRRAB9ALMNA
SCHEMBL2171155 0.74 SCN9A (0.52) SCN9AFPR2HTR1AHTR7DPP4
SCHEMBL11928250 0.73 ALDH1A1 (0.49) DPP4ALDH1A1TSHRHTTCYP3A4
SCHEMBL17220302 0.73 GAA (0.54) DPP4ALDH1A1TSHRRAB9ACYP3A4
SCHEMBL27828766 0.73 GAA (0.54) DPP4ALDH1A1TSHRRAB9ACYP3A4
SCHEMBL2172455 0.70 SCN9A (0.60) SCN9AFPR2HTR1AHTR7DPP4
SCHEMBL15797662 0.70 LMNA (0.54) ALDH1A1TSHRHTTCYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2349252-A2 SYNERGISTIC COMBINATION OF SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS AND ANTIMICROTUBULE AGENTS Exelixis, Inc. (US) 2011-08-03 EP disclosed