SCHEMBL21702046

SCHEMBL21702046

O=C(NC1CCCCC1)C(=O)C(C[C@@H]1CCNC1=O)NC(=O)[C@H](CC1CCCCC1)NC(=O)c1cc2ccccc2s1

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
REN P00797 1/20 0.45
CTSL P07711 2/20 0.44
CTSB P07858 2/20 0.44
OPRM1 P35372 1/20 0.42
CTSK P43235 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23506531 1.00 REN (0.45) RENCTSLCTSBOPRM1CTSK
SCHEMBL21702050 0.96 REN (0.44) RENCTSLCTSBOPRM1CTSK
SCHEMBL23506412 0.91 CTSL (0.45) RENCTSLCTSB
SCHEMBL23506296 0.91 CTSL (0.55) CTSLCTSBCTSK
SCHEMBL21702056 0.90 REN (0.46) RENCTSLCTSBOPRM1
SCHEMBL23506236 0.90 REN (0.46) RENCTSLCTSBOPRM1
SCHEMBL21702036 0.89 CTSL (0.47) RENCTSLCTSB
SCHEMBL23506499 0.89 CTSL (0.47) RENCTSLCTSB
SCHEMBL21702057 0.88 REN (0.44) RENCTSLCTSBOPRM1
SCHEMBL23506252 0.87 CTSK (0.51) CTSLCTSBCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021151387-A1 PHARMACEUTICAL USE OF KETOAMIDE-BASED COMPOUND 中国科学院上海药物研究所 2021-08-05 WO disclosed
WO-2020030143-A1 KETOAMIDE COMPOUND AND PREPARATION METHOD, PHARMACEUTICAL COMPOSITION, AND USE THEREOF 中国科学院上海药物研究所 2020-02-13 WO disclosed