SCHEMBL21702245

SCHEMBL21702245

O=C(CNC(=O)c1cc2ccccc2s1)NC(C[C@@H]1CCNC1=O)C(=O)C(=O)NC1CCCCC1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.47
CTSL P07711 1/20 0.41
CTSB P07858 1/20 0.41
CTSK P43235 1/20 0.37
TMIGD3 P0DMS9 1/20 0.36
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23506411 1.00 OPRM1 (0.47) OPRM1CTSLCTSBCTSKTMIGD3
SCHEMBL21702186 0.96 OPRM1 (0.47) OPRM1CTSLCTSBCTSKTMIGD3
SCHEMBL23506337 0.96 OPRM1 (0.47) OPRM1CTSLCTSBCTSKTMIGD3
SCHEMBL23506253 0.96 OPRM1 (0.47) OPRM1CTSLCTSBCTSKTMIGD3
SCHEMBL23506237 0.87 OPRM1 (0.43) OPRM1CTSLCTSBRAB9A
SCHEMBL23506251 0.87 OPRM1 (0.43) OPRM1CTSLCTSBRAB9A
SCHEMBL21702046 0.87 REN (0.45) OPRM1CTSLCTSBCTSK
SCHEMBL23506531 0.87 REN (0.45) OPRM1CTSLCTSBCTSK
SCHEMBL23506316 0.86 CTSL (0.45) OPRM1CTSLSLC6A2SLC6A4
SCHEMBL23711631 0.86 CTSL (0.45) OPRM1CTSLSLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020030143-A1 KETOAMIDE COMPOUND AND PREPARATION METHOD, PHARMACEUTICAL COMPOSITION, AND USE THEREOF 中国科学院上海药物研究所 2020-02-13 WO disclosed