SCHEMBL2170522

SCHEMBL2170522

CS(=O)(=O)c1cc(CCCN)cs1

nearest known ligand 0.34

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 1/20 0.33
CA2 P00918 9/20 0.33
LOX P28300 1/20 0.33
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24670388 0.69 CA2 (0.50) CA2
SCHEMBL24670395 0.69 CA2 (0.42) CA2
SCHEMBL6798039 0.67 CA2 (0.52) HTR6CA2TSHR
SCHEMBL28342951 0.66 DAO (0.44) TSHR
SCHEMBL25689016 0.66 HTR2A (0.46)
SCHEMBL2180225 0.65 CES2 (0.38) CA2
SCHEMBL15880882 0.64 CA2 (0.39) CA2
Hydrochloric Acid SCHEMBL1871819 0.63 CYP2A6 (0.41) CA2TSHR
SCHEMBL5215479 0.63 ENPP2 (0.38) CA2
SCHEMBL25689015 0.63 LTB4R (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346868-A1 AZAINDAZOLE COMPOUNDS AS CCR1 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-07-27 EP disclosed
WO-2010036632-A1 AZAINDAZOLE COMPOUNDS AS CCR1 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-04-01 WO disclosed