SCHEMBL21708618

SCHEMBL21708618

CCCC(F)OC(=O)CCBr

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.37
MAPT P10636 2/20 0.35
MAPK1 P28482 1/20 0.35
FAAH O00519 4/20 0.33
ALDH1A1 P00352 3/20 0.33
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33
CHRM1 P11229 1/20 0.32
AKR1A1 P14550 1/20 0.32
CHRM3 P20309 1/20 0.32
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
ADRA1A P35348 1/20 0.32
HRH1 P35367 1/20 0.32
DRD3 P35462 1/20 0.32
SLC6A3 Q01959 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC2 Q92769 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
CES2 O00748 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21708625 0.92 LMNA (0.43) LMNAMAPTMAPK1FAAHALDH1A1
SCHEMBL10525765 0.88 ALDH1A1 (0.46) LMNAMAPTMAPK1ALDH1A1CHRM1
SCHEMBL1933764 0.86 ALDH1A1 (0.41) LMNAMAPTFAAHALDH1A1CNR1
SCHEMBL3465881 0.79 CYP1A2 (0.48) LMNAMAPTMAPK1ALDH1A1HDAC1
SCHEMBL716434 0.76 CHRM1 (0.39) LMNAMAPTFAAHALDH1A1CHRM1
SCHEMBL3976804 0.76 MGAM (0.38) FAAHCNR1CNR2CHRM1AKR1A1
SCHEMBL4778558 0.76 FAAH (0.40) FAAHCNR1CNR2
SCHEMBL8816774 0.74 FFAR3 (0.44) LMNAALDH1A1HDAC1HDAC2TDP1
SCHEMBL28966490 0.74
SCHEMBL4300126 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3609870-A1 SUBSTITUTED N-ARYLETHYL-2-AMINOQUINOLINE-4-CARBOXAMIDES AND USE THEREOF Bayer Aktiengesellschaft (DE) 2020-02-19 EP disclosed
EP-3609869-A1 SUBSTITUTED N-ARYLETHYL-2-ARYLQUINOLINE-4-CARBOXAMIDES AND USE THEREOF Bayer Aktiengesellschaft (DE) 2020-02-19 EP disclosed