SCHEMBL21708905

SCHEMBL21708905

C#CCN(CC#C)CCc1cn(CC#C)c2ccc(O)cc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 6/20 0.39
HTR1D P28221 3/20 0.39
HTR1A P08908 2/20 0.39
HTR1B P28222 1/20 0.39
HTR1F P30939 1/20 0.39
HTR7 P34969 1/20 0.39
CYP19A1 P11511 1/20 0.36
PLA2G2A P14555 1/20 0.36
SPR P35270 1/20 0.33
ICMT O60725 1/20 0.32
ESR1 P03372 1/20 0.32
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA4 P22748 1/20 0.32
CA9 Q16790 1/20 0.32
MAOA P21397 1/20 0.31
MAOB P27338 1/20 0.31
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21709087 0.82 EGFR (0.42) HTR6HTR1DHTR1AHTR1BHTR1F
SCHEMBL21708936 0.81 HTR6 (0.42) HTR6BCHEMAPT
Hydrochloric Acid SCHEMBL21693918 0.81 EGFR (0.43) HTR6HTR1DHTR1AHTR1BHTR1F
SCHEMBL21708942 0.78 SPR (0.42) HTR6HTR1DHTR1AHTR1BHTR1F
SCHEMBL25057123 0.70 HTR1D (0.71) HTR6HTR1DHTR1AHTR1BHTR1F
SCHEMBL28672344 0.65 HTR6 (0.46) HTR6HTR1DHTR1AHTR1BHTR1F
SCHEMBL18602059 0.64 HTR6 (0.45) HTR6HTR1DHTR1AHTR1BHTR1F
SCHEMBL1120469 0.63 KCNH2 (0.38) HTR6
SCHEMBL21708941 0.62 ADRB2 (0.46) HTR6HTR1DHTR1AHTR1BMAOA
SCHEMBL21709100 0.62 MEN1 (0.33) HTR1DHTR2AMEN1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020032080-A1 COMPOUND, SALT OF COMPOUND, NEUROMODULATION AGENT, METHOD FOR EVALUATING NEUROMODULATION AGENT, METHOD FOR PRODUCING COMPOUND, AND METHOD FOR PRODUCING SALT OF COMPOUND 学校法人慶應義塾 2020-02-13 WO disclosed