SCHEMBL21709055

SCHEMBL21709055

C#CCOc1cc(C(CN)OCC#C)ccc1O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFKB1 P19838 1/20 0.41
BLM P54132 3/20 0.40
PMP22 Q01453 1/20 0.40
GAA P10253 2/20 0.36
HPGD P15428 4/20 0.34
MAPT P10636 3/20 0.34
APEX1 P27695 2/20 0.34
RECQL P46063 2/20 0.34
TDP1 Q9NUW8 2/20 0.34
CYP3A4 P08684 2/20 0.34
LMNA P02545 2/20 0.34
MEN1 O00255 1/20 0.34
ADRB2 P07550 1/20 0.34
ADRB1 P08588 1/20 0.34
ADRA2A P08913 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
ADRB3 P13945 1/20 0.34
DRD2 P14416 1/20 0.34
ADRA2B P18089 1/20 0.34
ADRA2C P18825 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21709063 0.87 MAOB (0.36) HPGDLMNAKMT2ATSHRMAOB
SCHEMBL21708869 0.85 TDP1 (0.49) NFKB1BLMPMP22HPGDMAPT
SCHEMBL21709056 0.83 NFKB1 (0.61) NFKB1BLMPMP22HPGDMAPT
SCHEMBL21709058 0.82 CYP3A4 (0.31) NFKB1CYP3A4TSHRHTR2A
SCHEMBL21709065 0.82 MAOA (0.40) NFKB1BLMPMP22GAAMAPT
SCHEMBL21709214 0.78
SCHEMBL21709245 0.76 P2RX3 (0.31) CGAS
SCHEMBL21709213 0.74 MAOB (0.30) MAOB
SCHEMBL21709064 0.72 TAAR1 (0.58) NFKB1BLMPMP22GAAMAPT
SCHEMBL21708896 0.71 NFKB1 (0.49) NFKB1BLMPMP22HPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020032080-A1 COMPOUND, SALT OF COMPOUND, NEUROMODULATION AGENT, METHOD FOR EVALUATING NEUROMODULATION AGENT, METHOD FOR PRODUCING COMPOUND, AND METHOD FOR PRODUCING SALT OF COMPOUND 学校法人慶應義塾 2020-02-13 WO disclosed