SCHEMBL21708896

SCHEMBL21708896

C#CCOc1ccc(C(O)CN)cc1OCC#C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFKB1 P19838 3/20 0.49
BLM P54132 5/20 0.48
PMP22 Q01453 3/20 0.48
TDP1 Q9NUW8 4/20 0.45
HPGD P15428 4/20 0.45
KDM4E B2RXH2 4/20 0.45
APEX1 P27695 3/20 0.45
MAPT P10636 3/20 0.45
RECQL P46063 3/20 0.45
TAAR1 Q96RJ0 3/20 0.45
LMNA P02545 3/20 0.45
MAPK1 P28482 2/20 0.45
ADRB2 P07550 2/20 0.45
ADRB1 P08588 2/20 0.45
ADRA2A P08913 2/20 0.45
ADRA2B P18089 2/20 0.45
ADRA2C P18825 2/20 0.45
ADRA1D P25100 2/20 0.45
MEN1 O00255 1/20 0.45
ADORA3 P0DMS8 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21709056 0.88 NFKB1 (0.61) NFKB1BLMPMP22TDP1HPGD
SCHEMBL21709063 0.80 MAOB (0.36) HPGDLMNAKMT2ATSHRMAOB
SCHEMBL21709053 0.80 KDM1A (0.40) NFKB1TDP1KDM4EMAPTRECQL
SCHEMBL7143077 0.79 NFKB1 (0.57) NFKB1BLMPMP22TDP1HPGD
SCHEMBL21709144 0.77 NFKB1 (0.41) NFKB1BLMPMP22TDP1HPGD
SCHEMBL21709155 0.77 NFKB1 (0.35) NFKB1BLMPMP22TDP1HPGD
SCHEMBL21708865 0.75 MAOB (0.33) BLMTDP1HPGDKDM4EAPEX1
SCHEMBL7148513 0.74 NFKB1 (0.48) NFKB1BLMPMP22TDP1HPGD
SCHEMBL9070525 0.74 NFKB1 (0.48) NFKB1BLMPMP22TDP1HPGD
SCHEMBL16774308 0.73 PPARG (0.51) DRD2KMT2AHIF1AMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020032080-A1 COMPOUND, SALT OF COMPOUND, NEUROMODULATION AGENT, METHOD FOR EVALUATING NEUROMODULATION AGENT, METHOD FOR PRODUCING COMPOUND, AND METHOD FOR PRODUCING SALT OF COMPOUND 学校法人慶應義塾 2020-02-13 WO disclosed