SCHEMBL21709099

SCHEMBL21709099

C#CCNCCc1c[nH]c2ccc(O)c(C#C)c12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 6/20 0.46
HTR2C P28335 4/20 0.39
KDM4E B2RXH2 3/20 0.39
MEN1 O00255 1/20 0.39
CYP2D6 P10635 1/20 0.39
KMT2A Q03164 1/20 0.39
KCNT1 Q5JUK3 1/20 0.37
HTR1A P08908 4/20 0.37
ALDH1A1 P00352 2/20 0.37
HTT P42858 1/20 0.37
HTR2B P41595 2/20 0.36
HTR7 P34969 2/20 0.36
HTR6 P50406 2/20 0.36
DRD1 P21728 1/20 0.36
HTR1D P28221 1/20 0.36
HTR1B P28222 1/20 0.36
HTR1E P28566 1/20 0.36
ADORA2A P29274 1/20 0.36
ADORA2B P29275 1/20 0.36
DRD3 P35462 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31708144 0.82 HTR2A (0.70) HTR2AHTR2CKDM4EMEN1KMT2A
SCHEMBL21709092 0.80 HTR2C (0.57) HTR2AHTR2CCYP2D6HTR1AHTR2B
SCHEMBL21709101 0.77 HTR1A (0.46) HTR2AHTR2CCYP2D6HTR1AHTR2B
SCHEMBL25057132 0.74 HTR2C (0.68) HTR2AHTR2CKDM4EMEN1CYP2D6
SCHEMBL26989205 0.72 HTR2A (0.70) HTR2AKDM4EMEN1KMT2AKCNT1
SCHEMBL21709102 0.72 KDM4E (0.42) HTR2AHTR2CKDM4EMEN1CYP2D6
SCHEMBL26989142 0.69 MTNR1A (0.60) HTR2AHTR2CHTR1AALDH1A1HTR2B
SCHEMBL31742959 0.69 HTR2A (0.68) HTR2AHTR2CKDM4EMEN1CYP2D6
SCHEMBL29206374 0.68 MPO (0.73) HTR2AKMT2AHTR1AMPOSLC6A4
SCHEMBL29992340 0.66 HTR2A (0.76) HTR2AHTR2CKDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020032080-A1 COMPOUND, SALT OF COMPOUND, NEUROMODULATION AGENT, METHOD FOR EVALUATING NEUROMODULATION AGENT, METHOD FOR PRODUCING COMPOUND, AND METHOD FOR PRODUCING SALT OF COMPOUND 学校法人慶應義塾 2020-02-13 WO disclosed