SCHEMBL21709263

SCHEMBL21709263

C#CCNCCc1cc(OC)c(OC)cc1C#C

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 16/20 0.42
HTR2C P28335 8/20 0.40
SMN1; SMN2 Q16637 1/20 0.39
HRH1 P35367 1/20 0.36
OPRM1 P35372 1/20 0.36
OPRK1 P41145 1/20 0.36
HTR2B P41595 1/20 0.36
HTR6 P50406 1/20 0.36
SLC2A1 P11166 1/20 0.36
ACHE P22303 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21708876 0.85 ACHE (0.34) HTR2AHTR2CACHE
SCHEMBL21709148 0.78 ACHE (0.35) HTR2AHTR2CACHE
SCHEMBL21708864 0.77 HTR2A (0.33) HTR2AHTR2CACHE
SCHEMBL21709091 0.77 TAAR1 (0.53) HTR2AHTR2C
SCHEMBL21709077 0.75 CA12 (0.43) HTR2AHTR2CSMN1; SMN2HTR2BACHE
SCHEMBL21709269 0.74 BCHE (0.39) HTR2AACHE
SCHEMBL21709074 0.73 ATM (0.63) SMN1; SMN2SLC2A1
SCHEMBL21709146 0.72 TSHR (0.36)
SCHEMBL21709262 0.69 P2RX3 (0.38) OPRM1
SCHEMBL2780581 0.67 SMN1; SMN2 (0.47) SMN1; SMN2ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020032080-A1 COMPOUND, SALT OF COMPOUND, NEUROMODULATION AGENT, METHOD FOR EVALUATING NEUROMODULATION AGENT, METHOD FOR PRODUCING COMPOUND, AND METHOD FOR PRODUCING SALT OF COMPOUND 学校法人慶應義塾 2020-02-13 WO disclosed