SCHEMBL21712430

SCHEMBL21712430

Nc1nc2cccc(O)c2c2c[nH]nc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.40
ACHE P22303 1/20 0.38
CHRM5 P08912 1/20 0.36
PDPK1 O15530 2/20 0.35
CCNT1 O60563 1/20 0.35
CCNB2 O95067 1/20 0.35
CDK1 P06493 1/20 0.35
HTR1A P08908 1/20 0.35
CCNB1 P14635 1/20 0.35
PRKACA P17612 1/20 0.35
CCNA2 P20248 1/20 0.35
PRKACG P22612 1/20 0.35
PRKACB P22694 1/20 0.35
CDK2 P24941 1/20 0.35
HTR2B P41595 1/20 0.35
GSK3B P49841 1/20 0.35
CDK9 P50750 1/20 0.35
CCNA1 P78396 1/20 0.35
CDK5 Q00535 1/20 0.35
SLC6A3 Q01959 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3991824 0.82 PARP1 (0.40) ACHEPDPK1NCF1DCPSTLR8
SCHEMBL21712387 0.79 DCPS (0.54) ACHEHTR1AHTR2BMAPTALDH1A1
SCHEMBL29526654 0.76 ADORA3 (0.47) ACHEMAPTGAAALDH1A1RAB9A
SCHEMBL1233223 0.76 ADORA3 (0.47) ACHEMAPTGAAALDH1A1RAB9A
SCHEMBL3990704 0.75 TLR7 (0.41) HTR2BDCPSDHFRTLR8TLR7
Hydrochloric Acid SCHEMBL5572086 0.74 ADORA3 (0.46) ACHEMAPTGAAALDH1A1RAB9A
Hydrochloric Acid SCHEMBL3995097 0.73 TLR8 (0.45) TLR8TLR7
SCHEMBL5568387 0.72 KCNH2 (0.33) TLR8TLR7
Hydrochloric Acid SCHEMBL5572201 0.72 KCNH2 (0.32) TLR8TLR7
SCHEMBL23421716 0.71 ACHE (0.39) ACHEGAAALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11834448-B2 2-amino-quinoline derivatives BIRDIE BIOPHARMACEUTICALS, INC. (KY) 2023-12-05 US claimed
EP-3615539-B1 2-AMINO-QUINOLINE DERIVATIVES BIRDIE BIOPHARMACEUTICALS INC (KY) 2023-08-09 EP claimed
US-20200055851-A1 2-AMINO-QUINOLINE DERIVATIVES BIRDIE BIOPHARMACEUTICALS, INC. (KY) 2020-02-20 US claimed
CN-110637018-A 2-amino-quinoline derivatives 博笛生物科技有限公司 2019-12-31 CN claimed
US-11834448-B2 2-amino-quinoline derivatives BIRDIE BIOPHARMACEUTICALS, INC. (KY) 2023-12-05 US disclosed
US-11834448-B2 2-amino-quinoline derivatives BIRDIE BIOPHARMACEUTICALS, INC. (KY) 2023-12-05 US disclosed
US-11834448-B2 2-amino-quinoline derivatives BIRDIE BIOPHARMACEUTICALS, INC. (KY) 2023-12-05 US disclosed
EP-3615539-B1 2-AMINO-QUINOLINE DERIVATIVES BIRDIE BIOPHARMACEUTICALS INC (KY) 2023-08-09 EP disclosed
EP-3615539-B1 2-AMINO-QUINOLINE DERIVATIVES BIRDIE BIOPHARMACEUTICALS INC (KY) 2023-08-09 EP disclosed
US-11053240-B2 2-amino-quinoline derivatives BIRDIE BIOPHARMACEUTICALS, INC. (KY) 2021-07-06 US disclosed
US-11053240-B2 2-amino-quinoline derivatives BIRDIE BIOPHARMACEUTICALS, INC. (KY) 2021-07-06 US disclosed
US-20200055851-A1 2-AMINO-QUINOLINE DERIVATIVES BIRDIE BIOPHARMACEUTICALS, INC. (KY) 2020-02-20 US disclosed
US-20200055851-A1 2-AMINO-QUINOLINE DERIVATIVES BIRDIE BIOPHARMACEUTICALS, INC. (KY) 2020-02-20 US disclosed
CN-110637018-A 2-amino-quinoline derivatives 博笛生物科技有限公司 2019-12-31 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11053240-B2 2-amino-quinoline derivatives TLR7, TLR8, TLR1 CYP1A2 1011/4885ACHE 3149/4885CHRM5 442/4885
US-20200055851-A1 2-AMINO-QUINOLINE DERIVATIVES TLR7, TLR8, TLR1 CYP1A2 1011/4885ACHE 3149/4885CHRM5 442/4885
US-11834448-B2 2-amino-quinoline derivatives TLR7, TLR8, TLR1 CYP1A2 1011/4885ACHE 3149/4885CHRM5 442/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.