SCHEMBL2171685

SCHEMBL2171685

Cc1ccc(-c2cc(C(=O)O[C@@H](C)C(N)=O)cc(-c3cc(C)ccc3C#N)c2)nc1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
S1PR3 Q99500 6/20 0.42
P2RX3 P56373 7/20 0.35
P2RX2 Q9UBL9 7/20 0.35
S1PR1 P21453 4/20 0.34
S1PR4 O95977 2/20 0.34
S1PR2 O95136 1/20 0.34
NR1I2 O75469 1/20 0.34
WNT3A P56704 1/20 0.33
PRMT5 O14744 1/20 0.33
WDR77 Q9BQA1 1/20 0.33
GRM5 P41594 1/20 0.33
XDH P47989 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2172000 0.87 S1PR3 (0.40) S1PR3P2RX3P2RX2S1PR1WNT3A
SCHEMBL2172263 0.85 NSD2 (0.37) S1PR3P2RX3P2RX2GRM5
SCHEMBL2170462 0.85 S1PR3 (0.41) S1PR3P2RX3P2RX2S1PR1NR1I2
SCHEMBL2173127 0.81 XDH (0.43) S1PR3P2RX3P2RX2WNT3AGRM5
SCHEMBL2171780 0.79 CYP11B2 (0.38) S1PR3WNT3AXDH
SCHEMBL2171503 0.79 P2RX3 (0.43) P2RX3P2RX2NR1I2
SCHEMBL2172981 0.79 P2RX3 (0.39) P2RX3P2RX2NR1I2
SCHEMBL2171681 0.77 P2RX3 (0.61) P2RX3P2RX2
SCHEMBL2170747 0.75 S1PR3 (0.40) S1PR3S1PR1NR1I2WNT3A
SCHEMBL2171994 0.73 P2RX3 (0.46) S1PR3P2RX3P2RX2S1PR1NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346825-A2 MODULATORS OF P2X3 RECEPTOR ACTIVITY Evotec AG (DE) 2011-07-27 EP disclosed