SCHEMBL2172263

SCHEMBL2172263

Cc1ccc(-c2cc(C(=O)O[C@@H](C)C(N)=O)cc(-c3ccc(C#N)cc3C)c2)nc1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NSD2 O96028 1/20 0.37
S1PR3 Q99500 1/20 0.37
GRM5 P41594 2/20 0.36
EGLN1 Q9GZT9 3/20 0.36
FPR2 P25090 1/20 0.36
SCN9A Q15858 1/20 0.36
OXTR P30559 3/20 0.36
CYP11B1 P15538 2/20 0.36
CYP11B2 P19099 2/20 0.36
MAP4K1 Q92918 1/20 0.35
P2RX3 P56373 2/20 0.35
P2RX2 Q9UBL9 2/20 0.35
AVPR1A P37288 2/20 0.35
SLC22A12 Q96S37 1/20 0.34
MAP4K4 O95819 1/20 0.34
MINK1 Q8N4C8 1/20 0.34
TNIK Q9UKE5 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2171685 0.85 S1PR3 (0.42) S1PR3GRM5P2RX3P2RX2
SCHEMBL3476174 0.82 GRM5 (0.43) NSD2GRM5EGLN1OXTRCYP11B1
SCHEMBL2170462 0.81 S1PR3 (0.41) S1PR3GRM5MAP4K1P2RX3P2RX2
SCHEMBL2172261 0.78 P2RX3 (0.59) P2RX3P2RX2
SCHEMBL2171503 0.77 P2RX3 (0.43) P2RX3P2RX2
SCHEMBL2172981 0.77 P2RX3 (0.39) CYP11B2P2RX3P2RX2
SCHEMBL2172000 0.73 S1PR3 (0.40) S1PR3P2RX3P2RX2
SCHEMBL2171780 0.72 CYP11B2 (0.38) S1PR3CYP11B2SLC22A12
SCHEMBL3474932 0.67 XDH (0.40) GRM5P2RX3P2RX2
SCHEMBL2171034 0.66 P2RX3 (0.39) P2RX3P2RX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346825-A2 MODULATORS OF P2X3 RECEPTOR ACTIVITY Evotec AG (DE) 2011-07-27 EP disclosed