SCHEMBL2172326

SCHEMBL2172326

CC(NC(=O)Cc1cnccn1)(C(N)=O)c1ccc(Oc2ccc(F)cc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RORC P51449 3/20 0.41
PTGER4 P35408 1/20 0.39
CYP3A4 P08684 1/20 0.37
MAPK14 Q16539 1/20 0.37
LMNA P02545 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
SCN9A Q15858 5/20 0.36
FPR2 P25090 2/20 0.36
BRD4 O60885 1/20 0.36
ACKR3 P25106 1/20 0.35
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34
KDM4E B2RXH2 1/20 0.34
KMT2A Q03164 1/20 0.34
ADRB1 P08588 1/20 0.33
ADRB3 P13945 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2357195 0.87 SCN9A (0.45) MAPK14LMNASMN1; SMN2SCN9ACA1
SCHEMBL2352914 0.84 CYP3A4 (0.48) RORCCYP3A4MAPK14LMNASMN1; SMN2
SCHEMBL2171613 0.78 EPHX2 (0.51) CYP3A4LMNASMN1; SMN2KDM4E
SCHEMBL2172340 0.74 SCN9A (0.51) SCN9AFPR2ADRB1ADRB3
SCHEMBL2172331 0.72 S1PR1 (0.52) SMN1; SMN2SCN9ABRD4KDM4EKMT2A
SCHEMBL2356374 0.72 MAPK14 (0.48) MAPK14
SCHEMBL2169794 0.70 ALDH1A1 (0.45) LMNASMN1; SMN2KDM4EKMT2A
SCHEMBL2172986 0.70 ALDH1A1 (0.40) CYP3A4LMNASMN1; SMN2KDM4EKMT2A
SCHEMBL2171604 0.70 SCN9A (0.44) LMNASMN1; SMN2SCN9AFPR2KDM4E
SCHEMBL2171837 0.70 ALDH1A1 (0.52) CYP3A4SCN9AFPR2KDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346821-A1 SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS Exelixis, Inc. (US) 2011-07-27 EP disclosed