SCHEMBL2352914

SCHEMBL2352914

CC(NC(=O)Cc1cccnc1)(C(N)=O)c1ccc(Oc2ccc(F)cc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.48
CYP1A2 P05177 1/20 0.48
CYP2C9 P11712 1/20 0.48
GAA P10253 1/20 0.47
MMP13 P45452 1/20 0.46
SCN9A Q15858 2/20 0.46
FAAH O00519 1/20 0.41
KDM4E B2RXH2 1/20 0.41
RORC P51449 5/20 0.41
GPR132 Q9UNW8 1/20 0.40
CDK9 P50750 1/20 0.40
MAPK8 P45983 1/20 0.40
LMNA P02545 2/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
HTT P42858 1/20 0.39
MAPK14 Q16539 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
NAMPT P43490 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2171613 0.87 EPHX2 (0.51) CYP3A4CYP2C9GAAKDM4ELMNA
SCHEMBL2172326 0.84 RORC (0.41) CYP3A4SCN9AKDM4ERORCLMNA
SCHEMBL2357195 0.80 SCN9A (0.45) SCN9ALMNAMAPTMAPK14SMN1; SMN2
SCHEMBL2356374 0.80 MAPK14 (0.48) MAPK14
SCHEMBL2352923 0.75 SCN9A (0.64) CYP3A4CYP1A2CYP2C9GAASCN9A
SCHEMBL11608799 0.73 KMT2A (0.51) CYP3A4GAAMMP13SCN9ALMNA
SCHEMBL2352920 0.72 S1PR1 (0.52) GAASCN9AKDM4ERORCLMNA
SCHEMBL2172986 0.72 ALDH1A1 (0.40) CYP3A4CYP1A2GAAMMP13KDM4E
SCHEMBL2757955 0.72 CYP1A2 (0.69) CYP3A4CYP1A2CYP2C9GAAKDM4E
SCHEMBL2171604 0.70 SCN9A (0.44) GAAMMP13SCN9AKDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2349252-A2 SYNERGISTIC COMBINATION OF SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS AND ANTIMICROTUBULE AGENTS Exelixis, Inc. (US) 2011-08-03 EP disclosed