SCHEMBL21731053

SCHEMBL21731053

CC1(C)OB(c2ccc3c(c2)OCO3)C1(C)C

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.39
TAAR1 Q96RJ0 3/20 0.38
ATM Q13315 1/20 0.38
POLB P06746 1/20 0.37
ALDH1A1 P00352 3/20 0.36
HSD17B10 Q99714 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
MAPK9 P45984 2/20 0.36
SLC6A4 P31645 3/20 0.35
SLC6A3 Q01959 3/20 0.35
MAPK1 P28482 1/20 0.35
SLC6A2 P23975 1/20 0.35
CMA1 P23946 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
MIF P14174 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30544472 0.79 LPL (0.44) CYP3A4ATMPOLBALDH1A1HSD17B10
SCHEMBL3148663 0.79 LPL (0.44) CYP3A4ATMPOLBALDH1A1HSD17B10
SCHEMBL5899518 0.73 POLB (0.40) CYP3A4TAAR1ATMPOLBALDH1A1
SCHEMBL15240051 0.70 RXRA (0.36) CYP3A4
SCHEMBL5899619 0.70 CYP3A4 (0.39) CYP3A4TAAR1ATMPOLBALDH1A1
SCHEMBL14212260 0.69 LPL (0.44) POLB
SCHEMBL29634547 0.69 LPL (0.44) POLB
SCHEMBL14746387 0.68 ALDH1A1 (0.55) POLBALDH1A1MAPK1MEN1KMT2A
SCHEMBL15241249 0.68 RXRA (0.34)
SCHEMBL30495575 0.68 TAAR1 (0.54) CYP3A4TAAR1SLC6A4SLC6A3SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3611174-A1 [1,2,4]TRIAZOLO[1,5-C]PYRIMIDINE DERIVATIVE AS A2A RECEPTOR INHIBITOR Medshine Discovery Inc. (CN) 2020-02-19 EP disclosed