SCHEMBL21732253

SCHEMBL21732253

CC(C)(C)OC(=O)N1Cc2cc(S(C)(=O)=O)ccc2[C@@H]1C(=O)Nc1cnc(N2CCC[C@@H]2c2cccc(F)c2)nc1

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
RORC P51449 19/20 0.47
CYP2D6 P10635 6/20 0.47
KCNH2 Q12809 1/20 0.47
IL17A Q16552 1/20 0.43
JAK2 O60674 1/20 0.42
NTRK1 P04629 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21732118 0.91 RORC (0.51) RORCCYP2D6KCNH2IL17A
SCHEMBL21732176 0.89 RORC (0.44) RORCCYP2D6KCNH2IL17AJAK2
SCHEMBL21732254 0.88 NTRK1 (0.41) JAK2NTRK1
SCHEMBL21732267 0.85 RORC (0.53) RORCCYP2D6KCNH2IL17A
SCHEMBL21732200 0.83 RORC (0.47) RORCCYP2D6KCNH2IL17A
SCHEMBL21732071 0.82 RORC (0.49) RORCJAK2NTRK1
SCHEMBL21732075 0.80 HDAC8 (0.38) RORCNTRK1
SCHEMBL21732280 0.80 RORC (0.56) RORCCYP2D6KCNH2IL17A
SCHEMBL21732119 0.79 NTRK1 (0.41) JAK2NTRK1
SCHEMBL21732235 0.78 RORC (0.50) RORCCYP2D6KCNH2IL17A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020035557-A1 NOVEL HETEROAROMATIC MODULATORS OF THE RETINOID-RELATED ORPHAN RECEPTOR GAMMA LEO PHARMA A/S (DK) 2020-02-20 WO disclosed