SCHEMBL21732235

SCHEMBL21732235

CC(=O)N1Cc2cc(S(C)(=O)=O)ccc2[C@@H]1C(=O)Nc1cnc(N2CC(F)(F)CC2c2cccc(F)c2)nc1

nearest known ligand 0.50

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
RORC P51449 20/20 0.50
CYP2D6 P10635 8/20 0.50
IL17A Q16552 1/20 0.50
KCNH2 Q12809 4/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21732232 0.89 NTRK1 (0.41) RORCCYP2D6IL17AKCNH2
SCHEMBL21732118 0.87 RORC (0.51) RORCCYP2D6IL17AKCNH2
SCHEMBL21732267 0.81 RORC (0.53) RORCCYP2D6IL17AKCNH2
SCHEMBL21732295 0.79 RORC (0.51) RORCCYP2D6IL17AKCNH2
SCHEMBL21732253 0.78 RORC (0.47) RORCCYP2D6IL17AKCNH2
SCHEMBL21732222 0.77 RORC (0.40) RORCCYP2D6IL17A
SCHEMBL21732119 0.76 NTRK1 (0.41)
SCHEMBL21732083 0.76 RORC (0.64) RORCCYP2D6IL17AKCNH2
SCHEMBL21732225 0.76 RORC (0.37) RORCCYP2D6IL17AKCNH2
SCHEMBL21732293 0.71 NTRK1 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020035557-A1 NOVEL HETEROAROMATIC MODULATORS OF THE RETINOID-RELATED ORPHAN RECEPTOR GAMMA LEO PHARMA A/S (DK) 2020-02-20 WO disclosed