SCHEMBL21732296

SCHEMBL21732296

CC(=O)N1Cc2cc([S+](C)[O-])ccc2C1C(=O)Nc1ccc(N2CC(C)CC2c2cccc(F)c2)nc1

nearest known ligand 0.37

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
RORC P51449 16/20 0.37
CYP2D6 P10635 11/20 0.37
IL17A Q16552 1/20 0.37
KCNH2 Q12809 4/20 0.37
JAK2 O60674 4/20 0.36
NTRK1 P04629 4/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21732225 0.92 RORC (0.37) RORCCYP2D6IL17AKCNH2JAK2
SCHEMBL21732198 0.91 NTRK1 (0.37) RORCCYP2D6KCNH2JAK2NTRK1
SCHEMBL21732220 0.88 NTRK1 (0.44) JAK2NTRK1
SCHEMBL21732295 0.88 RORC (0.51) RORCCYP2D6IL17AKCNH2
SCHEMBL21732285 0.86 JAK2 (0.35) RORCJAK2NTRK1
SCHEMBL21732119 0.81 NTRK1 (0.41) JAK2NTRK1
SCHEMBL21732232 0.80 NTRK1 (0.41) RORCCYP2D6IL17AKCNH2JAK2
SCHEMBL21732190 0.80 RORC (0.35) RORCCYP2D6IL17AKCNH2
SCHEMBL21732216 0.79 NTRK1 (0.44) JAK2NTRK1
SCHEMBL21732227 0.78 RORC (0.43) RORCCYP2D6IL17AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020035557-A1 NOVEL HETEROAROMATIC MODULATORS OF THE RETINOID-RELATED ORPHAN RECEPTOR GAMMA LEO PHARMA A/S (DK) 2020-02-20 WO disclosed