SCHEMBL2174025

SCHEMBL2174025

CC(C)(C)OC(=O)NC1CCN(C(=O)c2csc(CNC(=O)COc3ccc(OC(F)(F)F)cc3)n2)CC1.CC1CN(C(=O)c2csc(CNC(=O)COc3ccc(OC(F)(F)F)cc3)n2)CCN1c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.41
LIPE Q05469 1/20 0.38
ADORA2A P29274 5/20 0.36
ADORA2B P29275 4/20 0.36
ADORA3 P0DMS8 2/20 0.36
KDM5A P29375 1/20 0.36
NPC1L1 Q9UHC9 2/20 0.36
MCHR1 Q99705 2/20 0.35
EPHX2 P34913 2/20 0.35
CKS1B P61024 1/20 0.34
SKP1 P63208 1/20 0.34
SKP2 Q13309 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
TP53 P04637 1/20 0.34
NAMPT P43490 1/20 0.34
CHRM4 P08173 1/20 0.34
PARP1 P09874 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2174028 0.90 CHRM2 (0.37) CHRM2LIPEADORA2AADORA2BKDM5A
SCHEMBL5669978 0.84 CHRM2 (0.43) CHRM2LIPEMCHR1SMN1; SMN2TP53
SCHEMBL2174258 0.76 MCHR1 (0.40) MCHR1
SCHEMBL5668886 0.75 KMT2A (0.41) MCHR1EPHX2
SCHEMBL2173319 0.75 MCHR1 (0.40) MCHR1
SCHEMBL4387610 0.74 KDM4E (0.42) CHRM2MCHR1EPHX2SMN1; SMN2
SCHEMBL4389385 0.73 TAOK1 (0.43) MCHR1NAMPT
SCHEMBL4392436 0.73 POLB (0.53) CHRM2MCHR1EPHX2CHRM4
SCHEMBL5668976 0.72 LMNA (0.43) MCHR1EPHX2SMN1; SMN2
SCHEMBL5668246 0.72 L3MBTL1 (0.49) NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7973061-B2 Anaplastic lymphoma kinase modulators and methods of use EXELIXIS, INC. (US) 2011-07-05 US claimed