SCHEMBL2174028

SCHEMBL2174028

CC1CN(C(=O)c2csc(CNC(=O)C(CC(C)(C)OC(=O)NC3CCN(C(=O)c4csc(CNC(=O)COc5ccc(OC(F)(F)F)cc5)n4)CC3)Oc3ccc(OC(F)(F)F)cc3)n2)CCN1c1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.37
KDM5A P29375 2/20 0.34
LIPE Q05469 1/20 0.34
MCHR1 Q99705 3/20 0.32
EPHX2 P34913 4/20 0.32
TP53 P04637 2/20 0.31
PRKAA2 P54646 2/20 0.31
PRKAB2 O43741 1/20 0.31
PRKAG1 P54619 1/20 0.31
PRKAA1 Q13131 1/20 0.31
PRKAG3 Q9UGI9 1/20 0.31
PRKAG2 Q9UGJ0 1/20 0.31
PRKAB1 Q9Y478 1/20 0.31
GAA P10253 1/20 0.31
KCNH2 Q12809 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
CHRM4 P08173 1/20 0.30
LMNA P02545 1/20 0.30
ADORA2A P29274 2/20 0.30
ADORA2B P29275 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2174025 0.90 CHRM2 (0.41) CHRM2KDM5ALIPEMCHR1EPHX2
SCHEMBL5669978 0.79 CHRM2 (0.43) CHRM2LIPEMCHR1TP53SMN1; SMN2
SCHEMBL2174258 0.71 MCHR1 (0.40) MCHR1
SCHEMBL5668886 0.71 KMT2A (0.41) MCHR1EPHX2
SCHEMBL2173319 0.70 MCHR1 (0.40) MCHR1
SCHEMBL4387610 0.69 KDM4E (0.42) CHRM2MCHR1EPHX2GAASMN1; SMN2
SCHEMBL4389385 0.69 TAOK1 (0.43) MCHR1
SCHEMBL4392436 0.69 POLB (0.53) CHRM2MCHR1EPHX2PRKAA2PRKAB2
SCHEMBL5668976 0.68 LMNA (0.43) MCHR1EPHX2SMN1; SMN2LMNA
SCHEMBL5668246 0.67 L3MBTL1 (0.49) GAALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7973061-B2 Anaplastic lymphoma kinase modulators and methods of use EXELIXIS, INC. (US) 2011-07-05 US claimed