SCHEMBL21747449

SCHEMBL21747449

Nc1ccccc1-c1cc2ccc(CN3CCN(C(=O)O)CC3)cc2o1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 5/20 0.49
S1PR1 P21453 1/20 0.48
S1PR3 Q99500 1/20 0.48
GRIN2B Q13224 1/20 0.46
DRD2 P14416 4/20 0.46
FAAH O00519 1/20 0.43
MC4R P32245 1/20 0.42
MC5R P33032 1/20 0.42
DRD3 P35462 1/20 0.41
NR1H4 Q96RI1 1/20 0.41
NPC1 O15118 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30468227 0.85 SMARCA2 (0.43) DRD4S1PR1S1PR3GRIN2BDRD2
SCHEMBL21747470 0.84 FAAH (0.47) DRD4S1PR1S1PR3GRIN2BDRD2
SCHEMBL21747451 0.84 ALDH1A1 (0.49) DRD4S1PR1S1PR3DRD2NPC1
SCHEMBL20542002 0.82 MCHR1 (0.45) DRD4S1PR1S1PR3DRD2FAAH
SCHEMBL20541900 0.81 FAAH (0.50) DRD4S1PR1S1PR3FAAHNPC1
SCHEMBL20541620 0.80 S1PR1 (0.45) DRD4S1PR1S1PR3GRIN2BDRD2
SCHEMBL20541736 0.79 NPC1 (0.49) DRD4S1PR1S1PR3FAAHNPC1
SCHEMBL20541985 0.79 HDAC1 (0.49) DRD4S1PR1S1PR3FAAH
SCHEMBL20541721 0.79 KDM4E (0.52) DRD4S1PR1S1PR3FAAHMC4R
SCHEMBL21747444 0.79 S1PR1 (0.50) S1PR1S1PR3GRIN2BNR1H4NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3613735-B1 NOVEL SIRT 1 ACTIVATOR AND MEDICINAL USE THEREOF NAT UNIV PUSAN IND UNIV COOP FOUND (KR) 2023-04-12 EP disclosed
EP-3613735-A1 NOVEL SIRT 1 ACTIVATOR AND MEDICINAL USE THEREOF Pusan National University Industry - University Cooperation Foundation (KR) 2020-02-26 EP disclosed