SCHEMBL2175144

SCHEMBL2175144

CCCc1nc(N)cc(N)n1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.52
TDP1 Q9NUW8 1/20 0.52
NOS2 P35228 6/20 0.52
NOS3 P29474 4/20 0.52
NOS1 P29475 4/20 0.52
BACE1 P56817 1/20 0.38
HRH4 Q9H3N8 1/20 0.38
ADORA1 P30542 2/20 0.37
ADORA2A P29274 1/20 0.37
ADORA2B P29275 1/20 0.37
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
GFER P55789 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28330923 0.87 NOS2 (0.50) MAPTTDP1NOS2NOS3NOS1
SCHEMBL9378258 0.85 NOS2 (0.44) MAPTTDP1NOS2NOS3NOS1
SCHEMBL10344792 0.84 NOS2 (0.48) MAPTTDP1NOS2NOS3NOS1
SCHEMBL10830346 0.82 NOS2 (0.42) MAPTTDP1NOS2NOS3NOS1
SCHEMBL28267332 0.79 MAPT (0.56) MAPTTDP1NOS2NOS3NOS1
SCHEMBL29724038 0.75 MAPT (0.52) MAPTTDP1NOS2NOS3NOS1
SCHEMBL9521798 0.75 NOS2 (0.52) MAPTNOS2NOS3NOS1BACE1
SCHEMBL9738916 0.74 NOS2 (0.53) MAPTTDP1NOS2NOS3NOS1
SCHEMBL11811150 0.74 HRH4 (0.38) MAPTNOS2NOS3NOS1HRH4
SCHEMBL671139 0.74 CASP1 (0.62) NOS2NOS3NOS1HRH4ADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011079343-A2 SUBSTITUTED PYRIDINES AND PYRIMIDINES TECHNISCHE UNIVERSITAET WIEN (AT) 2011-07-07 WO claimed