SCHEMBL21753518

SCHEMBL21753518

NC(=O)C1=CN(c2ccc(F)cc2)C=CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
USP2 O75604 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
NPC1 O15118 3/20 0.34
RAB9A P51151 3/20 0.34
ALDH1A1 P00352 2/20 0.34
TP53 P04637 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
TSHR P16473 1/20 0.34
CASP1 P29466 1/20 0.34
CASP7 P55210 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
CA12 O43570 2/20 0.33
CA1 P00915 2/20 0.33
CA2 P00918 2/20 0.33
CA9 Q16790 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22092555 0.86 LDHA (0.33) MAPK1MEN1KMT2AALDH1A1KDM4E
SCHEMBL21753502 0.84 ALDH1A1 (0.35) SMN1; SMN2USP2RAB9AALDH1A1KDM4E
SCHEMBL21753524 0.84 ALDH1A1 (0.38) MAPK1SMN1; SMN2USP2MEN1KMT2A
SCHEMBL28854513 0.84 CA12 (0.38) SMN1; SMN2MEN1KMT2AALDH1A1KDM4E
SCHEMBL21891257 0.81 ALDH1A1 (0.45) MEN1KMT2ANPC1ALDH1A1MAPT
SCHEMBL21753516 0.77 TSHR (0.40) MAPK1SMN1; SMN2USP2MEN1KMT2A
SCHEMBL860052 0.74 PARP1 (0.44) ALDH1A1CCNA2CDK2CCNA1NOTUM
SCHEMBL1274356 0.67 LDHA (0.36) LDHA
SCHEMBL29217620 0.67 LDHA (0.34) LDHA
SCHEMBL28200009 0.64 LDHA (0.35) CCNA2CDK2CCNA1LDHA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020038460-A1 NOVEL QUINOLINE DERIVATIVE INHIBITOR 南京药捷安康生物科技有限公司 2020-02-27 WO disclosed