SCHEMBL21753550

SCHEMBL21753550

CCOC(=O)C(NNC1CC1)C(=O)/C(=C/N(C)C)c1ccc(F)cc1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
MAPT P10636 1/20 0.36
CASP3 P42574 1/20 0.36
TRPV1 Q8NER1 1/20 0.36
SENP7 Q9BQF6 1/20 0.36
EPHX2 P34913 5/20 0.35
PPARG P37231 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
ALDH1A1 P00352 1/20 0.35
TSHR P16473 1/20 0.34
FAAH O00519 1/20 0.34
CTSL P07711 1/20 0.34
THRB P10828 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21753551 1.00 CHRM1 (0.36) CHRM1MEN1KMT2AMAPTCASP3
SCHEMBL21753545 0.92 L3MBTL1 (0.36) MEN1KMT2AMAPTL3MBTL1TSHR
SCHEMBL21753508 0.87 RAB9A (0.37) EPHX2ALDH1A1FAAHCTSLNPC1
SCHEMBL21753506 0.87 RAB9A (0.37) EPHX2ALDH1A1FAAHCTSLNPC1
SCHEMBL21753556 0.79 NPC1 (0.38) MEN1KMT2AMAPTEPHX2ALDH1A1
SCHEMBL21753573 0.74 RAB9A (0.41) MEN1KMT2AMAPTEPHX2PPARG
SCHEMBL16109883 0.73 MAPT (0.51) MEN1KMT2AMAPTCASP3TRPV1
SCHEMBL16109884 0.73 MAPT (0.51) MEN1KMT2AMAPTCASP3TRPV1
SCHEMBL21769290 0.72 CHRM1 (0.38) CHRM1MEN1KMT2AMAPTCASP3
SCHEMBL30106507 0.72 CHRM1 (0.38) CHRM1MEN1KMT2AMAPTCASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020038460-A1 NOVEL QUINOLINE DERIVATIVE INHIBITOR 南京药捷安康生物科技有限公司 2020-02-27 WO disclosed