SCHEMBL2175545

SCHEMBL2175545

CC(C)(C)OC(=O)[C@H]1CCC(CNC2CC2)C[C@]1(C)C(=O)O

nearest known ligand 0.35

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.32
NPY2R P49146 1/20 0.31
KDM1A O60341 1/20 0.30
CTSS P25774 1/20 0.30
CTSK P43235 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2172483 0.76 CHRM2 (0.34)
SCHEMBL2174224 0.72 MAPK1 (0.30)
SCHEMBL2175191 0.69 USP2 (0.36) KMT2ACTSS
SCHEMBL2172712 0.68 HPGD (0.48) KMT2A
SCHEMBL25381609 0.67 BTK (0.47) KMT2AKDM1ACTSK
SCHEMBL31390565 0.67 KDM1A (0.34) KDM1A
Hydrochloric Acid SCHEMBL2172300 0.67
SCHEMBL2173732 0.65 GPR119 (0.36) KMT2AKDM1A
SCHEMBL2175295 0.65 MAPK1 (0.36) KMT2A
SCHEMBL2173780 0.64 CYP19A1 (0.35) KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9440958-B2 Substituted cyclic hydroxamates as inhibitors of matrix metalloproteinases INCYTE CORPORATION (US) 2016-09-13 US disclosed
US-20110224189-A1 SUBSTITUTED CYCLIC HYDROXAMATES AS INHIBITORS OF MATRIX METALLOPROTEINASES INCYTE CORPORATION 2011-09-15 US disclosed
US-7973041-B2 Antiarthritic agents; psoriasis; anticancer agents;antiallergens; metalloprotease inhibitors. INCYTE CORPORATION (US) 2011-07-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110224189-A1 SUBSTITUTED CYCLIC HYDROXAMATES AS INHIBITORS OF MATRIX METALLOPROTEINASES MMP25, MMP14, MMP9 KMT2A 1912/4885NPY2R 3904/4885KDM1A 697/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.