SCHEMBL21756889

SCHEMBL21756889

Cc1cc(C2CC2)ccc1Oc1ccc(N)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
TEAD4 Q15561 1/20 0.42
MAPT P10636 3/20 0.41
TDP1 Q9NUW8 2/20 0.41
POLB P06746 1/20 0.41
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
SLC6A3 Q01959 1/20 0.40
CYP3A4 P08684 1/20 0.39
TSHR P16473 1/20 0.39
MCHR1 Q99705 5/20 0.39
NCOA1 Q15788 1/20 0.38
NCOA3 Q9Y6Q9 1/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
MITF O75030 1/20 0.37
GAA P10253 1/20 0.37
GFER P55789 1/20 0.37
NLRP1 Q9C000 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23158861 0.85 ESR2 (0.41) ALDH1A1SMN1; SMN2TEAD4MAPTTDP1
SCHEMBL21765332 0.84 MAPT (0.45) ALDH1A1SMN1; SMN2TEAD4MAPTTDP1
SCHEMBL31457276 0.79 ALDH1A1 (0.55) ALDH1A1SMN1; SMN2TEAD4MAPTTDP1
SCHEMBL1155719 0.79 ALDH1A1 (0.55) ALDH1A1SMN1; SMN2TEAD4MAPTTDP1
SCHEMBL9076164 0.78 TEAD4 (0.41) ALDH1A1SMN1; SMN2TEAD4MAPTTDP1
SCHEMBL29510593 0.78 ALDH1A1 (0.59) ALDH1A1SMN1; SMN2TEAD4MAPTTDP1
SCHEMBL1810759 0.78 ALDH1A1 (0.59) ALDH1A1SMN1; SMN2TEAD4MAPTTDP1
SCHEMBL21756941 0.78 MAPT (0.45) ALDH1A1SMN1; SMN2MAPTTDP1POLB
SCHEMBL21770055 0.77 ALDH1A1 (0.61) ALDH1A1SMN1; SMN2TEAD4MAPTTDP1
SCHEMBL2992329 0.77 ALDH1A1 (0.52) ALDH1A1SMN1; SMN2TEAD4MAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020039088-A2 NOVEL COMPOUNDS Xeniopro GmbH (DE) 2020-02-27 WO disclosed
WO-2020039092-A2 NOVEL AROMATIC MOLECULES Xeniopro GmbH (DE) 2020-02-27 WO disclosed
US-9403829-B2 Pharmaceutical compositions of 7-(6-(2-hydroxypropan-2-yl)pyridin-3-yl)-1-((trans)-4-methoxycyclohexyl)-3,4-dihydropyrazino [2,3-b]pyrazin-2(1H)-one, a solid form thereof and methods of their use SIGNAL PHARMACEUTICALS, LLC (US) 2016-08-02 US disclosed