SCHEMBL21756912

SCHEMBL21756912

COC1(c2ccc(Oc3ccc(C45CC6CC(C4)C(C6)C5)cc3)cc2)CN(C)C1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.38
KMT2A Q03164 4/20 0.38
HTT P42858 2/20 0.38
RAD52 P43351 2/20 0.38
LMNA P02545 4/20 0.37
ALDH1A1 P00352 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.33
NPC1 O15118 1/20 0.33
HIF1A Q16665 3/20 0.32
CASP2 P42575 2/20 0.32
EPHX2 P34913 2/20 0.32
MAPT P10636 1/20 0.32
EPAS1 Q99814 1/20 0.31
CTSD P07339 3/20 0.31
BACE1 P56817 3/20 0.31
PRMT5 O14744 2/20 0.31
WDR77 Q9BQA1 2/20 0.31
BACE2 Q9Y5Z0 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27210042 0.93 MEN1 (0.43) MEN1KMT2AHTTRAD52LMNA
SCHEMBL27210046 0.77 LMNA (0.44) MEN1KMT2AHTTRAD52LMNA
SCHEMBL21756960 0.75 MEN1 (0.44) MEN1KMT2AHTTRAD52LMNA
SCHEMBL27845478 0.73 LMNA (0.61) MEN1KMT2AHTTRAD52LMNA
SCHEMBL16216731 0.70 LMNA (0.52) MEN1KMT2AHTTRAD52LMNA
SCHEMBL21756909 0.69 MEN1 (0.41) MEN1KMT2AHTTRAD52LMNA
SCHEMBL12040557 0.67 LMNA (0.57) MEN1KMT2ALMNAALDH1A1L3MBTL1
SCHEMBL21769895 0.67 LMNA (0.35) MEN1KMT2AHTTRAD52LMNA
SCHEMBL15055320 0.67 ALDH1A1 (0.79) MEN1KMT2ALMNAALDH1A1L3MBTL1
SCHEMBL19638852 0.67 ALDH1A1 (0.79) MEN1KMT2ALMNAALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020039092-A2 NOVEL AROMATIC MOLECULES Xeniopro GmbH (DE) 2020-02-27 WO disclosed
US-9403829-B2 Pharmaceutical compositions of 7-(6-(2-hydroxypropan-2-yl)pyridin-3-yl)-1-((trans)-4-methoxycyclohexyl)-3,4-dihydropyrazino [2,3-b]pyrazin-2(1H)-one, a solid form thereof and methods of their use SIGNAL PHARMACEUTICALS, LLC (US) 2016-08-02 US disclosed