SCHEMBL21756933

SCHEMBL21756933

CC(C)c1ccc(I)cc1N

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.41
GABRB1 P18505 1/20 0.41
GABRB2 P47870 1/20 0.41
SLC6A2 P23975 4/20 0.36
SLC6A4 P31645 4/20 0.36
TRPA1 O75762 1/20 0.34
LMNA P02545 1/20 0.34
CHRM1 P11229 1/20 0.34
ADRA1A P35348 1/20 0.34
HTR2B P41595 1/20 0.34
GAA P10253 2/20 0.33
SLC6A3 Q01959 2/20 0.33
POLB P06746 1/20 0.33
GFER P55789 1/20 0.33
ALDH1A1 P00352 1/20 0.33
ALOX12 P18054 1/20 0.33
HTT P42858 1/20 0.33
HIF1A Q16665 1/20 0.33
CFTR P13569 1/20 0.31
HSP90AA1 P07900 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4647387 0.84 GABRA1 (0.48) GABRA1GABRB1GABRB2SLC6A2SLC6A4
SCHEMBL12197671 0.78 GABRA1 (0.52) GABRA1GABRB1GABRB2SLC6A2TRPA1
SCHEMBL5486247 0.76 CASP1 (0.48) SLC6A2TRPA1LMNACHRM1ADRA1A
SCHEMBL49477 0.76 CASP1 (0.48) SLC6A2TRPA1LMNACHRM1ADRA1A
SCHEMBL16860570 0.76 GABRA1 (0.44) GABRA1GABRB1GABRB2SLC6A2TRPA1
SCHEMBL29368425 0.76 CASP1 (0.48) SLC6A2TRPA1LMNACHRM1ADRA1A
SCHEMBL3847726 0.74 TRPA1 (0.56) SLC6A2TRPA1LMNACHRM1ADRA1A
Hydrochloric Acid SCHEMBL11217552 0.74 CASP1 (0.46) SLC6A2TRPA1LMNACHRM1ADRA1A
SCHEMBL12224190 0.74 GABRA1 (0.43) GABRA1GABRB1GABRB2SLC6A2TRPA1
SCHEMBL2244195 0.74 ALDH1A1 (0.59) GABRA1GABRB2SLC6A2TRPA1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020039092-A2 NOVEL AROMATIC MOLECULES Xeniopro GmbH (DE) 2020-02-27 WO disclosed
WO-2020039094-A1 PHENOXY(HETERO)ARYL ETHERS OF ANTIPROLIFERATIVE ACTIVITY Xeniopro GmbH (DE) 2020-02-27 WO disclosed
WO-2020039088-A2 NOVEL COMPOUNDS Xeniopro GmbH (DE) 2020-02-27 WO disclosed
US-9403829-B2 Pharmaceutical compositions of 7-(6-(2-hydroxypropan-2-yl)pyridin-3-yl)-1-((trans)-4-methoxycyclohexyl)-3,4-dihydropyrazino [2,3-b]pyrazin-2(1H)-one, a solid form thereof and methods of their use SIGNAL PHARMACEUTICALS, LLC (US) 2016-08-02 US disclosed
CN-1069312-C Substituted imidogen sulfamide, its preparation, use and medicines containing the same HOECHST AG (DE) 2001-08-08 CN disclosed
CN-1155538-A Substituted imidogen sulfamide, its preparation, use and medicines containing the same HOECHST AG (DE) 1997-07-30 CN disclosed