SCHEMBL21756945

SCHEMBL21756945

CC(C)c1c(F)cc(I)cc1C#N

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 2/20 0.33
GABRA1 P14867 1/20 0.31
GABRB1 P18505 1/20 0.31
GABRB2 P47870 1/20 0.31
CYP11B1 P15538 4/20 0.31
CYP11B2 P19099 4/20 0.31
ADRB2 P07550 1/20 0.31
ADRB1 P08588 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13748207 0.81 TRPV4 (0.35) TRPV4CYP11B1CYP11B2ADRB2ADRB1
SCHEMBL21756924 0.80 GABRA1 (0.41) GABRA1GABRB1GABRB2
SCHEMBL24606679 0.79 ADRB2 (0.40) TRPV4GABRA1GABRB2CYP11B1CYP11B2
SCHEMBL26457748 0.79 CYP11B1 (0.35) TRPV4CYP11B1CYP11B2ADRB2ADRB1
SCHEMBL807520 0.79 TRPV4 (0.34) TRPV4CYP11B1CYP11B2ADRB2ADRB1
SCHEMBL18999982 0.79 TRPV4 (0.41) TRPV4CYP11B1CYP11B2ADRB2ADRB1
SCHEMBL26458345 0.78 KHK (0.36) TRPV4GABRA1GABRB1CYP11B1CYP11B2
SCHEMBL13748982 0.75 CYP11B1 (0.39) CYP11B1CYP11B2
SCHEMBL21765351 0.75 TRPV4 (0.36) TRPV4CYP11B1CYP11B2
SCHEMBL11960299 0.74 TRPV4 (0.31) TRPV4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020039092-A2 NOVEL AROMATIC MOLECULES Xeniopro GmbH (DE) 2020-02-27 WO disclosed
WO-2020039088-A2 NOVEL COMPOUNDS Xeniopro GmbH (DE) 2020-02-27 WO disclosed
WO-2020039094-A1 PHENOXY(HETERO)ARYL ETHERS OF ANTIPROLIFERATIVE ACTIVITY Xeniopro GmbH (DE) 2020-02-27 WO disclosed