SCHEMBL21756947

SCHEMBL21756947

CNCc1cc(I)cc(F)c1C(C)C

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 5/20 0.32
KCNH2 Q12809 4/20 0.32
HTR2A P28223 3/20 0.32
SLC6A2 P23975 1/20 0.31
MCL1 Q07820 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21756926 0.79 GABRA1 (0.35)
SCHEMBL21756927 0.79 GABRA1 (0.31)
SCHEMBL21756924 0.77 GABRA1 (0.41)
SCHEMBL21756932 0.76 ALDH1A1 (0.38) SLC6A4HTR2ASLC6A2
SCHEMBL21756925 0.76 PRKCE (0.33)
SCHEMBL21765352 0.74 SLC6A4 (0.33) SLC6A4KCNH2HTR2ASLC6A2MCL1
SCHEMBL21756930 0.70 GABRA1 (0.35) MCL1
SCHEMBL21765276 0.70 GABRA1 (0.35)
SCHEMBL21769673 0.68 GABRA1 (0.34)
SCHEMBL21765277 0.68 GABRA1 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020039092-A2 NOVEL AROMATIC MOLECULES Xeniopro GmbH (DE) 2020-02-27 WO disclosed
WO-2020039088-A2 NOVEL COMPOUNDS Xeniopro GmbH (DE) 2020-02-27 WO disclosed
WO-2020039094-A1 PHENOXY(HETERO)ARYL ETHERS OF ANTIPROLIFERATIVE ACTIVITY Xeniopro GmbH (DE) 2020-02-27 WO disclosed
US-9403829-B2 Pharmaceutical compositions of 7-(6-(2-hydroxypropan-2-yl)pyridin-3-yl)-1-((trans)-4-methoxycyclohexyl)-3,4-dihydropyrazino [2,3-b]pyrazin-2(1H)-one, a solid form thereof and methods of their use SIGNAL PHARMACEUTICALS, LLC (US) 2016-08-02 US disclosed